SCHEMBL14966331

SCHEMBL14966331

O=C(CN1CCOc2nc([N+](=O)[O-])cn2CC1)NCCc1cccc(C(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
POLB P06746 2/20 0.42
MAPT P10636 3/20 0.42
TAAR1 Q96RJ0 1/20 0.40
ALDH1A1 P00352 3/20 0.37
CNR1 P21554 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
PARP1 P09874 1/20 0.36
DPP4 P27487 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NAMPT P43490 1/20 0.36
CCR1 P32246 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966262 0.92 POLB (0.49) LMNAKMT2APOLBMAPTALDH1A1
SCHEMBL14966138 0.87 NAMPT (0.43) LMNAMEN1KMT2AALDH1A1PARP1
SCHEMBL14966065 0.85 LMNA (0.54) LMNAMEN1KMT2APOLBMAPT
SCHEMBL14966242 0.84 LMNA (0.44) LMNAMEN1KMT2APOLBMAPT
SCHEMBL14965968 0.84 LMNA (0.48) LMNAALDH1A1CNR1KDM4E
SCHEMBL14966219 0.83 CA1 (0.48) KMT2APOLBMAPTALDH1A1
SCHEMBL14965849 0.80 CHRM1 (0.44) POLB
SCHEMBL14965644 0.80 CA1 (0.46) LMNAKMT2APOLBALDH1A1
SCHEMBL14966114 0.78 KCNH2 (0.38) LMNAPOLBMAPTALDH1A1KDM4E
SCHEMBL14965599 0.78 KDM4E (0.45) LMNAKMT2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed