SCHEMBL14966592

SCHEMBL14966592

O=C(O)c1cc(CCc2ccccc2)[nH]c(=O)c1

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 13/20 0.67
KDM5A P29375 1/20 0.48
KDM5B Q9UGL1 1/20 0.48
DAO P14920 3/20 0.46
GAA P10253 1/20 0.44
BACE1 P56817 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6613866 0.85 SMN1; SMN2 (0.57) GPR84KDM5AKDM5BDAO
SCHEMBL14967358 0.84 GPR84 (0.58) GPR84
SCHEMBL6695551 0.79 GPR84 (0.69) GPR84DAOBACE1
SCHEMBL8885796 0.78 MPO (0.51) GPR84KDM5AKDM5B
SCHEMBL11858938 0.78 GPR84 (0.68) GPR84DAOBACE1
SCHEMBL3676992 0.75 GPR84 (0.55) GPR84
SCHEMBL27766830 0.75 GAA (0.59) DAOGAA
SCHEMBL14603936 0.75 HCAR2 (0.54) GPR84KDM5BDAO
SCHEMBL3672125 0.74 ALDH1A1 (0.37) GPR84
SCHEMBL56627 0.74 ALDH1A1 (0.44) GPR84DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780014-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF Constellation Pharmaceuticals, Inc. (US) 2014-09-24 EP disclosed
WO-2013075083-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2013-05-23 WO disclosed