SCHEMBL14966620

SCHEMBL14966620

Cc1cc(C)c(CNC(=O)c2ccc(CCOCC(C)C)cc2)c(O)n1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 5/20 0.41
MAP4K1 Q92918 2/20 0.38
NR1H4 Q96RI1 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
RAB9A P51151 2/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
ESRRG P62508 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
EZH2 Q15910 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
USP2 O75604 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966453 0.89 NR1H4 (0.39) KLKB1MAP4K1NR1H4SMN1; SMN2RAB9A
SCHEMBL14966634 0.88 TSHR (0.42) KLKB1MAP4K1NR1H4SMN1; SMN2OPRM1
SCHEMBL14966830 0.87 KLKB1 (0.44) KLKB1MAP4K1NR1H4SMN1; SMN2OPRM1
SCHEMBL14966778 0.82 NPC1 (0.49) SMN1; SMN2ALDH1A1NPC1POLBMAPT
SCHEMBL14966659 0.82 LMNA (0.48) KLKB1SMN1; SMN2RAB9ANPC1MEN1
SCHEMBL14966459 0.82 KLKB1 (0.40) KLKB1MAP4K1NR1H4SMN1; SMN2MEN1
SCHEMBL14966781 0.82 RAB9A (0.47) KLKB1NR1H4SMN1; SMN2RAB9AALDH1A1
SCHEMBL14966619 0.81 EZH2 (0.40) KLKB1MAP4K1SMN1; SMN2OPRM1OPRK1
SCHEMBL14966647 0.81 SCN9A (0.44) SMN1; SMN2RAB9AALDH1A1MAPTHPGD
SCHEMBL14966474 0.81 MAPK14 (0.44) SMN1; SMN2RAB9AALDH1A1NPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780013-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF Constellation Pharmaceuticals, Inc. (US) 2014-09-24 EP disclosed
WO-2013075084-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2013-05-23 WO disclosed