SCHEMBL14966634

SCHEMBL14966634

Cc1cc(C)c(CNC(=O)c2ccc(CCOC(C)C)cc2)c(O)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KLKB1 P03952 3/20 0.42
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAP4K1 Q92918 1/20 0.39
NR1H4 Q96RI1 2/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
HTT P42858 1/20 0.38
EZH2 Q15910 1/20 0.38
PAX8 Q06710 1/20 0.38
MMP10 P09238 1/20 0.37
MMP8 P22894 1/20 0.37
MMP13 P45452 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
ESRRG P62508 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966830 0.89 KLKB1 (0.44) KLKB1ALDH1A1MEN1KMT2AMAP4K1
SCHEMBL14966620 0.88 KLKB1 (0.41) KLKB1ALDH1A1MEN1KMT2AMAP4K1
SCHEMBL14966453 0.86 NR1H4 (0.39) L3MBTL1KLKB1KMT2AMAP4K1NR1H4
SCHEMBL14966659 0.83 LMNA (0.48) KLKB1MEN1KMT2ASMN1; SMN2NPC1
SCHEMBL14966778 0.83 NPC1 (0.49) ALDH1A1SMN1; SMN2HTTMMP13NPC1
SCHEMBL14966459 0.83 KLKB1 (0.40) KLKB1MEN1KMT2AMAP4K1NR1H4
SCHEMBL14966781 0.83 RAB9A (0.47) TSHRKLKB1ALDH1A1NR1H4SMN1; SMN2
SCHEMBL14967113 0.82 LMNA (0.50) TSHRL3MBTL1SMN1; SMN2HTTMMP13
SCHEMBL14966647 0.82 SCN9A (0.44) ALDH1A1SMN1; SMN2MMP13RAB9A
SCHEMBL14966474 0.82 MAPK14 (0.44) L3MBTL1ALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780013-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF Constellation Pharmaceuticals, Inc. (US) 2014-09-24 EP disclosed
WO-2013075084-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2013-05-23 WO disclosed