SCHEMBL14967362

SCHEMBL14967362

O=C(O)c1c[nH]c(=O)n(CCc2ccc(F)cc2)c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.42
ALDH1A1 P00352 3/20 0.41
MITF O75030 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HDAC1 Q13547 3/20 0.40
HDAC11 Q96DB2 3/20 0.40
HDAC8 Q9BY41 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HAT1 O14929 1/20 0.39
EP300 Q09472 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL459138 0.73 KDM4E (0.38) ALDH1A1MAPTKMT2AKDM4E
SCHEMBL14969067 0.73 MEN1 (0.53) ALDH1A1HTTSMN1; SMN2MAPTMEN1
SCHEMBL10823654 0.71 PDE4A (0.38) ALDH1A1HTTMEN1KMT2AKDM4E
SCHEMBL6238938 0.70 KMT2A (0.56) ALDH1A1HTTRAB9ASMN1; SMN2HDAC1
SCHEMBL31198448 0.70 KMT2A (0.48) ALDH1A1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL16863377 0.69 PPARA (0.37) KDM4E
SCHEMBL10823648 0.68 B3GNT2 (0.46) ALDH1A1SMN1; SMN2KMT2AKDM4ECYP3A4
SCHEMBL425896 0.68 SLC9A1 (0.35) ALDH1A1KMT2AKDM4E
SCHEMBL14967295 0.68 KDM4E (0.39) ALDH1A1HTTRAB9ASMN1; SMN2MAPT
SCHEMBL10208376 0.67 KDM5A (0.48) DAOALDH1A1MITFHTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780338-A1 URACIL DERIVATIVES AS AXL AND C-MET KINASE INHIBITORS Cephalon, Inc. (US) 2014-09-24 EP disclosed
WO-2013074633-A1 URACIL DERIVATIVES AS AXL AND C-MET KINASE INHIBITORS CEPHALON, INC. (US) 2013-05-23 WO disclosed