SCHEMBL6238938

SCHEMBL6238938

O=C(O)c1ccc2[nH]c(=O)n(CCc3ccc(F)cc3)c(=O)c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.56
MEN1 O00255 3/20 0.56
ALDH1A1 P00352 7/20 0.51
GAA P10253 6/20 0.51
HSD17B10 Q99714 5/20 0.51
KDM4E B2RXH2 4/20 0.51
HPGD P15428 3/20 0.51
MAPT P10636 5/20 0.48
RXFP1 Q9HBX9 2/20 0.48
POLB P06746 2/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
KCNH2 Q12809 2/20 0.47
RAB9A P51151 1/20 0.47
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
HTR1A P08908 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020296 0.90 MAPT (0.57) KMT2AMEN1ALDH1A1GAAHSD17B10
SCHEMBL7634269 0.89 ALDH1A1 (0.49) KMT2AMEN1ALDH1A1GAAHSD17B10
SCHEMBL6431684 0.88 MAPT (0.52) ALDH1A1GAAHSD17B10KDM4EHPGD
SCHEMBL7012169 0.86 ALDH1A1 (0.47) KMT2AMEN1ALDH1A1GAAHSD17B10
SCHEMBL7019254 0.85 ALDH1A1 (0.48) KMT2AMEN1ALDH1A1GAAHSD17B10
SCHEMBL7052320 0.85 PTPN5 (0.55) KMT2AMEN1ALDH1A1GAAHSD17B10
SCHEMBL7620889 0.79 HPGD (0.47) KMT2AMEN1ALDH1A1GAAHSD17B10
SCHEMBL4252528 0.79 CACNA1G (0.63) KMT2AMEN1ALDH1A1GAAHSD17B10
SCHEMBL7191192 0.78 ALDH1A1 (0.60) KMT2AMEN1ALDH1A1GAAHSD17B10
SCHEMBL6218489 0.78 HPGD (0.65) KMT2AMEN1ALDH1A1GAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1531904-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 THAT IS NOT CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-25 EP disclosed
WO-2004007024-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 THAT IS NOT CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed