SCHEMBL14967862

SCHEMBL14967862

COC(=O)C12CCC(Oc3ncc(-c4ccc(C=O)c(F)c4)cn3)(CC1)CC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 6/20 0.39
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32
GRIN2B Q13224 2/20 0.32
ABL1 P00519 2/20 0.31
HDAC8 Q9BY41 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HDAC4 P56524 1/20 0.31
PIK3CG P48736 2/20 0.31
PIK3CD O00329 1/20 0.31
EGFR P00533 1/20 0.31
HCK P08631 1/20 0.31
SRC P12931 1/20 0.31
KDR P35968 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14967786 0.77 ERN1 (0.45) ERN1
SCHEMBL14967566 0.73 ERN1 (0.47) ERN1ALDH1A1MAPTPDGFRBPDGFRA
SCHEMBL14968320 0.72 HSD11B1 (0.35) MAPTKDM4EMEN1KMT2A
SCHEMBL15245235 0.71 DGAT1 (0.41) ERN1ALDH1A1MAPT
SCHEMBL14969513 0.70 ALDH1A1 (0.40) ERN1ALDH1A1MAPTGRIN2BKDM4E
SCHEMBL14969514 0.70 ALDH1A1 (0.40) ERN1ALDH1A1MAPTGRIN2BKDM4E
SCHEMBL14968063 0.70 ALDH1A1 (0.39) ERN1ALDH1A1MAPTGRIN2BKDM4E
SCHEMBL14968064 0.69 ALDH1A1 (0.40) ERN1ALDH1A1MAPTGRIN2BKDM4E
SCHEMBL14968031 0.69 ERN1 (0.46) ERN1GRIN2BABL1PIK3CGPIK3CD
SCHEMBL14967450 0.67 ERN1 (0.35) ERN1ALDH1A1MAPTGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed
WO-2013074387-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2013-05-23 WO disclosed