SCHEMBL14969448

SCHEMBL14969448

O=[N+]([O-])c1cn2c(n1)OCCN(Cc1cccc(-c3ccc4cc[nH]c4c3)c1)CC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
GFER P55789 1/20 0.41
KMT2A Q03164 1/20 0.41
TNIK Q9UKE5 2/20 0.39
MAPK14 Q16539 1/20 0.38
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38
BACE1 P56817 1/20 0.37
DHODH Q02127 1/20 0.36
FAAH O00519 1/20 0.36
FGFR1 P11362 1/20 0.36
FGFR2 P21802 1/20 0.36
FGFR3 P22607 1/20 0.36
KDR P35968 1/20 0.36
PRKACA P17612 4/20 0.36
PRKACG P22612 4/20 0.36
PRKACB P22694 4/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14971085 0.94 TNIK (0.40) MEN1GAAGFERKMT2ATNIK
SCHEMBL14971091 0.87 DRD2 (0.44) MEN1GAAKMT2AFAAHDRD2
SCHEMBL14969428 0.86 MAP3K11 (0.42) TNIKMAPK14PIK3CAMTORFAAH
SCHEMBL14966205 0.85 LSS (0.46) DRD2DRD4DRD3KDM4EALDH1A1
SCHEMBL14966131 0.85 DRD2 (0.49) MEN1GAAKMT2ADRD2DRD4
SCHEMBL14965795 0.83 CYP11B1 (0.45) DRD2DRD4DRD3
SCHEMBL14966240 0.83 KIT (0.40) TNIKDRD2DRD4DRD3
SCHEMBL14966336 0.82 DRD2 (0.45) TNIKFAAHADORA2AADORA1DRD2
SCHEMBL14966082 0.81 FAAH (0.46) MEN1KMT2ADHODHFAAHKDM4E
SCHEMBL14966085 0.81 FAAH (0.46) MEN1KMT2ADHODHFAAHKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed