SCHEMBL14969428

SCHEMBL14969428

O=[N+]([O-])c1cn2c(n1)OCCN(Cc1ccc(-c3ccc4[nH]ccc4c3)cc1)CC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 7/20 0.42
FLT1 P17948 2/20 0.42
MAPK14 Q16539 2/20 0.42
TNIK Q9UKE5 2/20 0.42
SGK1 O00141 1/20 0.42
IKBKB O14920 1/20 0.42
AURKA O14965 1/20 0.42
CHUK O15111 1/20 0.42
PRKAB2 O43741 1/20 0.42
ROCK2 O75116 1/20 0.42
ABL1 P00519 1/20 0.42
NTRK1 P04629 1/20 0.42
INSR P06213 1/20 0.42
LCK P06239 1/20 0.42
CDK1 P06493 1/20 0.42
IGF1R P08069 1/20 0.42
MET P08581 1/20 0.42
CYP3A4 P08684 1/20 0.42
SRC P12931 1/20 0.42
CDK2 P24941 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14971085 0.92 TNIK (0.40) FLT1MAPK14TNIKAURKBEGFR
SCHEMBL14969448 0.86 MEN1 (0.41) MAPK14TNIKPIK3CAMTORPRKCQ
SCHEMBL14971108 0.84 ALDH1A1 (0.44) FAAHALDH1A1LMNAMAPTKCNJ1
SCHEMBL14965513 0.83 LSS (0.46) ALDH1A1LMNAMAPTKCNJ1SMN1; SMN2
SCHEMBL14965918 0.82 ALDH1A1 (0.37) KCNH2JAK2ALDH1A1LMNAMAPT
SCHEMBL14965746 0.82 DRD2 (0.41) KCNH2DRD4ALDH1A1LMNAMAPT
SCHEMBL14966014 0.81 CHRNA7 (0.42) KCNH2LRRK2FAAHCHEK1ALDH1A1
SCHEMBL14965626 0.81 LTA4H (0.40) MAPK1FAAHALDH1A1LMNAMAPT
SCHEMBL14965511 0.81 LTA4H (0.40) MAPK1FAAHALDH1A1LMNAMAPT
SCHEMBL14966198 0.81 KCNJ1 (0.40) AURKAALDH1A1LMNAMAPTKCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed