SCHEMBL14972716

SCHEMBL14972716

Cn1c(=O)c2c(S(C)(=O)=O)snc2n(C)c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ADORA2A P29274 5/20 0.36
ALDH1A1 P00352 3/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MLKL Q8NB16 1/20 0.35
ADORA2B P29275 3/20 0.34
PIK3CD O00329 2/20 0.34
ADORA3 P0DMS8 2/20 0.34
ADORA1 P30542 2/20 0.34
POLB P06746 1/20 0.34
CNR1 P21554 1/20 0.34
ACHE P22303 1/20 0.34
NTSR1 P30989 1/20 0.34
MC3R P41968 1/20 0.34
NOTUM Q6P988 1/20 0.34
SIRT3 Q9NTG7 1/20 0.34
GDA Q9Y2T3 1/20 0.34
NR2E1 Q9Y466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9972885 0.71 KDM4E (0.41) KDM4EADORA2AALDH1A1ADORA2BKMT2A
SCHEMBL9972908 0.71 KMT2A (0.44) KDM4EADORA2AALDH1A1HSD17B10ADORA2B
SCHEMBL1689509 0.71 KDM4E (0.47) KDM4EADORA2AALDH1A1ADORA2BPIK3CD
SCHEMBL1689535 0.67 ADORA2B (0.40) KDM4EADORA2AALDH1A1CASP1CASP7
SCHEMBL3716133 0.67 ADORA2B (0.38) KDM4EADORA2AALDH1A1ADORA2BPIK3CD
SCHEMBL13190508 0.66 ALOX15 (0.42) KDM4EALDH1A1ADORA2BMAPT
SCHEMBL21602606 0.66 MLKL (0.58) ADORA2AALDH1A1MLKLADORA2BKMT2A
SCHEMBL14981101 0.64 ALDH1A1 (0.36) KDM4EALDH1A1POLBKMT2ARXFP1
SCHEMBL21602497 0.63 ADORA2A (0.40) KDM4EADORA2AALDH1A1CASP1CASP7
SCHEMBL475287 0.63 ADORA2B (0.37) KDM4EALDH1A1ADORA2BPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411397-B1 ISOTHIAZOLO-PYRIMIDINEDIONE DERIVATIVES AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS SA (CH) 2013-05-29 EP disclosed