SCHEMBL15025645

SCHEMBL15025645

COc1cc(C2CCN(C(=O)O)CC2)ncn1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.41
MAPK7 Q13164 7/20 0.40
PROKR1 Q8TCW9 1/20 0.38
TRPC6 Q9Y210 4/20 0.38
CYP2C19 P33261 1/20 0.38
CYP17A1 P05093 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
QDPR P09417 1/20 0.36
CSNK2A2 P19784 1/20 0.36
CSNK2A1 P68400 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14991022 0.83 HTT (0.51) MEN1KMT2A
SCHEMBL25465007 0.80 CYP2C19 (0.41) KMOCYP2C19CYP17A1
SCHEMBL10323271 0.80 KMO (0.45) KMOMAPK7PROKR1TRPC6CYP17A1
SCHEMBL17613226 0.80 CYP2C19 (0.41) KMOMAPK7PROKR1TRPC6CYP2C19
SCHEMBL21597925 0.78 HTR1A (0.53) MAPK7MEN1KMT2ALMNA
SCHEMBL25791777 0.77 KMO (0.44) KMOPROKR1CYP2C19CYP17A1
SCHEMBL1557826 0.76 GPR119 (0.49)
SCHEMBL15191875 0.75 TRPC6 (0.48) TRPC6
SCHEMBL14990759 0.73 HTR2C (0.41) CYP2C19MEN1KMT2A
SCHEMBL22143097 0.72 PIK3CD (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013083741-A1 1,2,4 -TRIAZOLES AS ALLOSTERIC MODULATORS OF MGLU5 RECEPTOR ACTIVITY FOR THE TREATMENT OF SCHIZOPHRENIA OF DEMENTIA BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-13 WO disclosed