SCHEMBL1503082

SCHEMBL1503082

COc1ccc(Cc2cc(C(N)=O)cnc2C(N)=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.51
VNN1 O95497 3/20 0.50
PARP10 Q53GL7 2/20 0.47
PARP1 P09874 2/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
PARP2 Q9UGN5 1/20 0.47
PARP4 Q9UKK3 1/20 0.47
CHEK2 O96017 1/20 0.46
MAP4K4 O95819 1/20 0.46
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
NNMT P40261 1/20 0.42
POLB P06746 1/20 0.41
NR3C2 P08235 1/20 0.41
SAE1 Q9UBE0 1/20 0.40
UBA2 Q9UBT2 1/20 0.40
APP P05067 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29567644 0.79 VNN1 (0.55) HPGDSVNN1PARP10PARP1CA1
SCHEMBL29056033 0.78 GRM2 (0.47) PARP10PARP1CA1CA2PARP2
SCHEMBL27858247 0.77 CYP19A1 (0.47) CA1CA2CHEK2POLB
SCHEMBL27915062 0.77 PARP10 (0.56) VNN1PARP10PARP1CA1CA2
SCHEMBL28349713 0.77 PARP10 (0.56) VNN1PARP10PARP1CA1CA2
SCHEMBL30478243 0.75 NNMT (0.41) HPGDSPARP10PARP1NNMT
SCHEMBL8213818 0.75 PARP10 (0.78) VNN1PARP10PARP1CA1CA2
SCHEMBL28285907 0.75 NNMT (0.41) HPGDSPARP10PARP1NNMT
SCHEMBL28127922 0.74 PARP10 (0.59) VNN1PARP10PARP1CA1CA2
SCHEMBL4001952 0.74 PARP10 (0.56) VNN1PARP10PARP1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300433-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE Ambrilia Biopharma Inc. (CA) 2011-03-30 EP disclosed