SCHEMBL15034067

SCHEMBL15034067

COc1cccc(C(=O)N2CCN(C(=O)c3ncn(-c4cccc(Cl)c4)n3)C(C)(C)C2)c1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.47
ALDH1A1 P00352 4/20 0.45
HPGD P15428 1/20 0.45
ABL1 P00519 4/20 0.44
BCR P11274 4/20 0.44
MGLL Q99685 2/20 0.43
WNK1 Q9H4A3 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
CCKAR P32238 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15034093 0.96 WNK1 (0.47) GRM5ALDH1A1HPGDABL1BCR
SCHEMBL15034139 0.92 ALDH1A1 (0.47) ALDH1A1HPGDABL1BCRL3MBTL1
SCHEMBL15019972 0.92 SLC6A7 (0.43) GRM5ALDH1A1HPGDMGLL
SCHEMBL15034043 0.90 MAPT (0.41) GRM5ALDH1A1HPGDMGLLDRD2
SCHEMBL15034061 0.90 MGLL (0.45) GRM5HPGDMGLL
SCHEMBL15034096 0.89 GRM5 (0.38) GRM5ALDH1A1HPGDMGLL
SCHEMBL15020006 0.88 ALDH1A1 (0.44) GRM5ALDH1A1HPGDL3MBTL1
SCHEMBL15034064 0.88 CCKAR (0.41) GRM5ALDH1A1HPGDMGLLWNK1
SCHEMBL15034036 0.88 ALDH1A1 (0.44) GRM5ALDH1A1HPGDMGLL
SCHEMBL15034215 0.88 HPGD (0.43) GRM5ALDH1A1HPGDMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8883789-B2 Piperazine derivatives and their use as positive allosteric modulators of mGluR5 receptors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-11 US disclosed
US-8883789-B2 Piperazine derivatives and their use as positive allosteric modulators of mGluR5 receptors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-11 US disclosed
US-20130158042-A1 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-20 US disclosed
US-20130158042-A1 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130158042-A1 NOVEL COMPOUNDS GRM5, GRIK5, GRM1 GRM5 1/4885ALDH1A1 3952/4885HPGD 2696/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.