SCHEMBL15037433

SCHEMBL15037433

CN(C)c1ccc(S(=O)(=O)Nc2ccc(I)cc2[N+](=O)[O-])cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.53
NFE2L2 Q16236 1/20 0.53
ALDH3A1 P30838 1/20 0.53
CA9 Q16790 1/20 0.50
MAPT P10636 6/20 0.49
ALDH1A1 P00352 6/20 0.49
TDP1 Q9NUW8 4/20 0.48
NPSR1 Q6W5P4 1/20 0.47
LMNA P02545 3/20 0.45
MAPK1 P28482 1/20 0.45
GFER P55789 1/20 0.45
MCL1 Q07820 1/20 0.45
CHEK1 O14757 1/20 0.44
AURKA O14965 1/20 0.44
JAK2 O60674 1/20 0.44
ABL1 P00519 1/20 0.44
NTRK1 P04629 1/20 0.44
CSF1R P07333 1/20 0.44
RET P07949 1/20 0.44
MET P08581 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15009060 0.85 ALDH1A1 (0.57) KEAP1NFE2L2ALDH3A1CA9MAPT
SCHEMBL28704611 0.84 MAPT (0.64) CA9MAPTALDH1A1TDP1LMNA
SCHEMBL15009245 0.73 MAPT (0.51) CA9MAPTALDH1A1TDP1NPSR1
SCHEMBL6364323 0.72 MAPT (0.50) ALDH3A1MAPTALDH1A1NPSR1KMT2A
SCHEMBL14676341 0.71 HCAR3 (0.58) MAPTALDH1A1TDP1LMNAMAPK1
SCHEMBL6553223 0.71 MAPT (0.59) MAPTALDH1A1TDP1LMNAKDR
SCHEMBL28186748 0.71 MAPT (0.54) MAPTALDH1A1TDP1LMNACRHBP
SCHEMBL21708265 0.70 MAPT (0.62) KEAP1NFE2L2ALDH3A1MAPTALDH1A1
SCHEMBL2006238 0.70 MAPT (0.72) KEAP1NFE2L2CA9MAPTALDH1A1
SCHEMBL30557374 0.70 MAPT (0.72) KEAP1NFE2L2CA9MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013090227-A1 BENZISOTHIAZOL-3(1H)-ONE-5-SULFONYL DERIVATIVES AS CHEMOKINE RECEPTOR MODULATORS ALLERGAN, INC. (US) 2013-06-20 WO disclosed