SCHEMBL1504840

SCHEMBL1504840

C[C@](CNC(=O)c1ccc(OCc2ccc(F)cc2)cc1)(C(=O)O)N1CCN(S(C)(=O)=O)CC1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 7/20 0.61
CHRM4 P08173 1/20 0.48
NR4A2 P43354 1/20 0.45
POLB P06746 1/20 0.45
MAOB P27338 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
BCL2L1 Q07817 1/20 0.43
MCL1 Q07820 1/20 0.43
SLC6A5 Q9Y345 1/20 0.43
PARP10 Q53GL7 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1504934 0.92 ADAM17 (0.63) ADAM17MAOBSLC6A5ALDH1A1
SCHEMBL1504974 0.92 ADAM17 (0.60) ADAM17MAOBKMT2AMEN1LMNA
SCHEMBL1504939 0.92 ADAM17 (0.60) ADAM17POLBKMT2AMEN1ALDH1A1
SCHEMBL1504779 0.92 ADAM17 (0.61) ADAM17CHRM4KMT2AMEN1HDAC1
SCHEMBL10276029 0.85 ADAM17 (0.61) ADAM17CHRM4NR4A2POLBMAOB
SCHEMBL1504684 0.82 ALDH1A1 (0.42) ADAM17POLBKMT2AMEN1ALDH1A1
SCHEMBL1504784 0.81 ADAM17 (0.43) ADAM17POLBALDH1A1
SCHEMBL1504797 0.81 ADAM17 (0.60) ADAM17ALDH1A1
SCHEMBL1504530 0.81 ADAM17 (0.60) ADAM17ALDH1A1
SCHEMBL1504967 0.79 ADAM17 (0.65) ADAM17ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011033009-A1 N- [2-HYDROXYCARBAMOYL-2- (PIPERAZINYL) ETHYL] BENZAMIDE COMPOUNDS, THEIR PREPARATION AND THEIR USE AS TACE INHIBITORS GALDERMA RESEARCH & DEVELOPMENT (FR) 2011-03-24 WO disclosed