SCHEMBL1504784

SCHEMBL1504784

COCCOCOc1ccc(C(=O)NC[C@@](C)(C(=O)O)N2CCN(S(C)(=O)=O)CC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 12/20 0.43
ALDH1A1 P00352 2/20 0.43
ADAM10 O14672 1/20 0.41
MMP3 P08254 1/20 0.41
ADAM9 Q13443 1/20 0.41
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
POLB P06746 1/20 0.38
HRH2 P25021 1/20 0.38
HRH1 P35367 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1504823 0.90 ALDH1A1 (0.41) ADAM17ALDH1A1TP53MAPTPOLB
SCHEMBL1503623 0.87 ALDH1A1 (0.46) ADAM17ALDH1A1TP53POLB
SCHEMBL1503650 0.85 ALDH1A1 (0.59) ALDH1A1TP53POLB
SCHEMBL1504825 0.85 ALDH1A1 (0.45) ADAM17ALDH1A1MAPTPOLBHRH2
SCHEMBL1504939 0.84 ADAM17 (0.60) ADAM17ALDH1A1TP53MAPTPOLB
SCHEMBL1504779 0.84 ADAM17 (0.61) ADAM17ADAM10MMP3
SCHEMBL1504797 0.83 ADAM17 (0.60) ADAM17ALDH1A1ADAM10MMP3ADAM9
SCHEMBL1504530 0.83 ADAM17 (0.60) ADAM17ALDH1A1ADAM10MMP3ADAM9
SCHEMBL1504974 0.82 ADAM17 (0.60) ADAM17ALDH1A1ADAM10MMP3MAPT
SCHEMBL1504684 0.82 ALDH1A1 (0.42) ADAM17ALDH1A1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011033009-A1 N- [2-HYDROXYCARBAMOYL-2- (PIPERAZINYL) ETHYL] BENZAMIDE COMPOUNDS, THEIR PREPARATION AND THEIR USE AS TACE INHIBITORS GALDERMA RESEARCH & DEVELOPMENT (FR) 2011-03-24 WO disclosed