SCHEMBL15048620

SCHEMBL15048620

Cn1nc(-c2ccc3ccccc3n2)cc1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 11/20 0.49
NPC1 O15118 10/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
NCF1 P14598 2/20 0.48
NOS2 P35228 1/20 0.48
BACE1 P56817 1/20 0.48
KDM4E B2RXH2 7/20 0.47
ALDH1A1 P00352 7/20 0.47
SMN1; SMN2 Q16637 5/20 0.47
MAPT P10636 4/20 0.47
TP53 P04637 4/20 0.47
HSD17B10 Q99714 4/20 0.47
PKM P14618 3/20 0.47
HPGD P15428 3/20 0.47
CYP3A4 P08684 2/20 0.47
THPO P40225 2/20 0.47
GMNN O75496 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15048619 0.79 NPC1 (0.46) RAB9ANPC1MEN1KMT2ANCF1
SCHEMBL29374931 0.75 RAB9A (0.64) RAB9ANPC1MEN1KMT2ANCF1
SCHEMBL170196 0.75 RAB9A (0.64) RAB9ANPC1MEN1KMT2ANCF1
SCHEMBL31749169 0.73 ADORA2B (0.38) RAB9ANPC1MEN1KMT2AKDM4E
SCHEMBL30883993 0.73 RAB9A (0.61) RAB9ANPC1MEN1KMT2ANCF1
Hydrochloric Acid SCHEMBL31243061 0.73 ALDH1A1 (0.63) RAB9ANPC1MEN1KMT2ANCF1
SCHEMBL34463709 0.73 RAB9A (0.61) RAB9ANPC1MEN1KMT2ANCF1
SCHEMBL10866984 0.73 RAB9A (0.61) RAB9ANPC1MEN1KMT2ANCF1
SCHEMBL31365172 0.73 RAB9A (0.61) RAB9ANPC1MEN1KMT2ANCF1
SCHEMBL31490600 0.73 RAB9A (0.61) RAB9ANPC1MEN1KMT2ANCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2526098-B1 NITROGEN-CONTAINING HETEROARYL DERIVATIVES HOFFMANN LA ROCHE (CH) 2018-07-11 EP claimed
US-8470820-B2 Nitrogen-containing heteroaryl derivatives HOFFMAN-LA ROCHE INC. (US) 2013-06-25 US claimed
EP-2526098-B1 NITROGEN-CONTAINING HETEROARYL DERIVATIVES HOFFMANN LA ROCHE (CH) 2018-07-11 EP disclosed
US-8470820-B2 Nitrogen-containing heteroaryl derivatives HOFFMAN-LA ROCHE INC. (US) 2013-06-25 US disclosed