SCHEMBL15054523

SCHEMBL15054523

COc1ccc(N(CC(=O)C(C)C)C(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RNF4 P78317 1/20 0.49
ALDH1A1 P00352 2/20 0.47
TSHR P16473 1/20 0.45
KEAP1 Q14145 2/20 0.44
NFE2L2 Q16236 2/20 0.44
BCL2A1 Q16548 2/20 0.43
LDHA P00338 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.42
LMNA P02545 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
TSPO P30536 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15053613 0.81 CYP3A4 (0.45) ALDH1A1BCL2A1TRPM8
SCHEMBL5702218 0.78 RNF4 (0.51) RNF4ALDH1A1TSHRKEAP1NFE2L2
SCHEMBL17628547 0.78 RNF4 (0.58) RNF4ALDH1A1TSHRKEAP1NFE2L2
SCHEMBL1429908 0.77 RNF4 (0.45) RNF4ALDH1A1TSHRKEAP1NFE2L2
SCHEMBL7044788 0.76 TSHR (0.51) RNF4ALDH1A1TSHRKEAP1NFE2L2
SCHEMBL15054037 0.75 LTB4R2 (0.50) RNF4TSHRKEAP1NFE2L2BCL2A1
SCHEMBL249712 0.74 RNF4 (0.48) RNF4ALDH1A1TSHRBCL2A1TRPM8
SCHEMBL11482380 0.73 OPRM1 (0.42) RNF4ALDH1A1TSHRBCL2A1TRPM8
SCHEMBL7106756 0.72 KEAP1 (0.55) RNF4TSHRKEAP1NFE2L2KMT2A
SCHEMBL1337080 0.72 USP2 (0.60) RNF4ALDH1A1TSHRBCL2A1TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013095301-A1 METHOD OF PREPARING CHIRAL KETONES FROM ALDEHYDES NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2013-06-27 WO disclosed