SCHEMBL15055355

SCHEMBL15055355

CS(=O)(=O)Nc1ccccc1Cc1ccc(Br)cc1F

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
NR3C1 P04150 6/20 0.42
PGR P06401 1/20 0.40
NR3C2 P08235 1/20 0.40
AR P10275 1/20 0.40
SLC22A12 Q96S37 1/20 0.40
TOP2A P11388 1/20 0.39
TOP2B Q02880 1/20 0.39
PSIP1 O75475 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KEAP1 Q14145 1/20 0.38
PTGS1 P23219 1/20 0.38
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15055390 0.79 ALDH1A1 (0.46) ALDH1A1NR3C1L3MBTL1KEAP1PTGS1
SCHEMBL23703126 0.78 NR3C1 (0.56) ALDH1A1NR3C1PGRNR3C2AR
SCHEMBL7160434 0.78 NR3C1 (0.43) ALDH1A1NR3C1PGRNR3C2AR
SCHEMBL26697138 0.77 NPC1 (0.48) ALDH1A1L3MBTL1KMT2A
SCHEMBL30526897 0.76 KMT2A (0.56) ALDH1A1SLC22A12L3MBTL1KMT2A
SCHEMBL2350815 0.76 KMT2A (0.56) ALDH1A1SLC22A12L3MBTL1KMT2A
SCHEMBL4157469 0.73 SLC22A12 (0.50) ALDH1A1SLC22A12PTGS1KMT2A
SCHEMBL3970765 0.72 NR3C1 (0.81) NR3C1PGRNR3C2AR
SCHEMBL13172655 0.72 P2RX7 (0.45)
SCHEMBL31500466 0.71 SLC22A12 (0.49) ALDH1A1NR3C1SLC22A12KEAP1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2793873-A1 BENZYL SULFONAMIDE DERIVATIVES AS RORc MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2014-10-29 EP disclosed
EP-2794584-A1 BENZYL SULFONAMIDE DERIVATIVES AS RORc MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2014-10-29 EP disclosed
WO-2013092941-A1 BENZYL SULFONAMIDE DERIVATIVES AS RORc MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2013-06-27 WO disclosed
WO-2013092939-A1 BENZYL SULFONAMIDE DERIVATIVES AS RORc MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2013-06-27 WO disclosed