SCHEMBL15062706

SCHEMBL15062706

COc1ccc2c(c1)c(C(=O)c1nnc(-c3ccccn3)o1)c(C)n2Cc1ccnc(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 11/20 0.50
ALDH1A1 P00352 3/20 0.45
PKM P14618 1/20 0.45
TSHR P16473 2/20 0.44
PLA2G1B P04054 1/20 0.43
POLB P06746 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HTT P42858 1/20 0.42
MAPT P10636 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005111 0.92 PLA2G2A (0.57) PLA2G2AALDH1A1PKMTSHRPLA2G1B
SCHEMBL2002769 0.92 PLA2G2A (0.52) PLA2G2AALDH1A1PKMTSHRPLA2G1B
SCHEMBL2006942 0.91 PLA2G2A (0.50) PLA2G2AALDH1A1PKMTSHRPLA2G1B
SCHEMBL2006756 0.89 PTGS2 (0.51) PLA2G2AALDH1A1TSHRPLA2G1BKMT2A
SCHEMBL3003525 0.87 PLA2G2A (0.47) PLA2G2AALDH1A1PKMTSHRPLA2G1B
SCHEMBL2002529 0.85 PLA2G2A (0.43) PLA2G2AALDH1A1PKMTSHRPLA2G1B
SCHEMBL2006833 0.84 PLA2G2A (0.44) PLA2G2AALDH1A1PKMTSHRPLA2G1B
SCHEMBL2005823 0.82 ALDH1A1 (0.52) PLA2G2AALDH1A1PKMTSHRPLA2G1B
SCHEMBL2002690 0.82 FAAH (0.50) PLA2G2AALDH1A1PKMTSHRMEN1
SCHEMBL2002857 0.82 ALDH1A1 (0.50) PLA2G2AALDH1A1PKMTSHRPLA2G1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2610244-A1 Indole compounds Ironwood Pharmaceuticals, Inc. (US) 2013-07-03 EP disclosed