SCHEMBL15071874

SCHEMBL15071874

COc1c(C)c(C)c(OC)c(Cc2c(C)c(OC)c(C)c(C)c2OC)c1C

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.42
CA4 P22748 2/20 0.42
CA1 P00915 1/20 0.42
CA6 P23280 1/20 0.42
IMPDH2 P12268 6/20 0.33
IMPDH1 P20839 1/20 0.32
CNR2 P34972 1/20 0.30
GPR55 Q9Y2T6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919191 0.86 CA2 (0.44) CA2CA4CA1CA6IMPDH2
SCHEMBL3044602 0.79 IMPDH2 (0.31) CA2CA4CA1CA6IMPDH2
SCHEMBL2029504 0.79 IMPDH2 (0.33) CA2CA4CA1CA6IMPDH2
SCHEMBL7508538 0.79 CA2 (0.34) CA2CA4CA1CA6IMPDH2
SCHEMBL9549629 0.79 CA2 (0.46) CA2CA4IMPDH2IMPDH1
SCHEMBL9310576 0.79 CNR2 (0.49) CNR2GPR55
SCHEMBL2952712 0.78 ACHE (0.40) CA2CA4CA1CA6
SCHEMBL9309164 0.77 LTA4H (0.50) CA2CA1
SCHEMBL1783169 0.75 HTR2A (0.46) IMPDH2IMPDH1
SCHEMBL1820953 0.75 IMPDH2 (0.32) IMPDH2IMPDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9770515-B2 Crosslinking of proteins and other entities via conjugates of α-haloacetophenones, benzyl halides, quinones, and their derivatives ADVANCED PROTEOME THERAPEUTICS INC. (US) 2017-09-26 US disclosed
US-20130165382-A1 CROSSLINKING OF PROTEINS AND OTHER ENTITIES VIA CONJUGATES OF ALPHA-HALOACETOPHENONES, BENZYL HALIDES, QUINONES, AND THEIR DERIVATIVES ADVANCED PROTEOME THERAPEUTICS INC. (US) 2013-06-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130165382-A1 CROSSLINKING OF PROTEINS AND OTHER ENTITIES VIA CONJUGATES OF ALPHA-HALOACETOPHENONES, BENZYL HALIDES, QUINONES, AND THEIR DERIVATIVES TBCA, HSP90AB2P, HSP90B1 CA2 2962/4885CA4 2988/4885CA1 3166/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.