SCHEMBL15079353

SCHEMBL15079353

COc1ccc2nccc(-c3cnc(OC)c(Cl)c3)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 4/20 0.49
TLR8 Q9NR97 2/20 0.48
KDM4E B2RXH2 2/20 0.46
MAPK1 P28482 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
LMNA P02545 1/20 0.45
HTR1A P08908 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
KCNH2 Q12809 1/20 0.41
GRM4 Q14833 1/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
CYP17A1 P05093 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
NCF1 P14598 1/20 0.41
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26420650 0.86 TLR8 (0.60) AAK1TLR8KDM4EMAPK1NPSR1
SCHEMBL15056707 0.81 PRKCZ (0.47)
SCHEMBL15056708 0.81 PRKCZ (0.47)
SCHEMBL10157305 0.76 PIK3CA (0.57) TLR8KDM4EMAPK1NPSR1LMNA
SCHEMBL30440258 0.76 PIK3CA (0.57) TLR8KDM4EMAPK1NPSR1LMNA
SCHEMBL282245 0.76 LMNA (0.58) KDM4EMAPK1NPSR1LMNAHTR1A
SCHEMBL29729443 0.76 LMNA (0.58) KDM4EMAPK1NPSR1LMNAHTR1A
SCHEMBL2051073 0.75 MAP3K14 (0.57) TLR8KDM4EMAPK1NPSR1LMNA
SCHEMBL13191354 0.70 TLR8 (0.65) TLR8KDM4EMAPK1NPSR1LMNA
SCHEMBL12988592 0.70 TLR8 (0.58) TLR8KDM4EMAPK1NPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013093850-A1 QUINOLINE DERIVATIVES NOVARTIS AG (CH) 2013-06-27 WO disclosed