SCHEMBL282245

SCHEMBL282245

COc1ccc2nccc(Cl)c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.58
KDM4E B2RXH2 2/20 0.56
HTR1A P08908 3/20 0.55
ADRA1D P25100 3/20 0.55
ADRA1A P35348 3/20 0.55
ADRA1B P35368 3/20 0.55
MAPK1 P28482 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
NCF1 P14598 1/20 0.51
MTNR1A P48039 3/20 0.51
MTNR1B P49286 3/20 0.51
RIPK2 O43353 2/20 0.50
CYP1A2 P05177 1/20 0.50
GAK O14976 1/20 0.50
COQ8A Q8NI60 1/20 0.50
NLK Q9UBE8 1/20 0.50
KDR P35968 1/20 0.48
ROCK2 O75116 1/20 0.46
CCR1 P32246 1/20 0.46
CCR5 P51681 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29729443 1.00 LMNA (0.58) LMNAKDM4EHTR1AADRA1DADRA1A
SCHEMBL201122 0.86 HTR1A (0.58) LMNAKDM4EHTR1AADRA1DADRA1A
SCHEMBL29362202 0.86 HTR1A (0.58) LMNAKDM4EHTR1AADRA1DADRA1A
SCHEMBL28581110 0.81 LMNA (0.61) LMNAKDM4EHTR1AADRA1DADRA1A
SCHEMBL1496335 0.80 LMNA (0.59) LMNAKDM4EHTR1AADRA1DADRA1A
SCHEMBL28810851 0.79 MTNR1A (0.49) LMNAKDM4EMAPK1NPSR1MTNR1A
SCHEMBL11767672 0.79 LMNA (0.58) LMNAKDM4EHTR1AADRA1DADRA1A
SCHEMBL18544268 0.79 KDM4E (0.60) LMNAKDM4EHTR1AADRA1DADRA1A
SCHEMBL591852 0.79 LMNA (0.62) LMNAKDM4EHTR1AADRA1DADRA1A
SCHEMBL590225 0.79 LMNA (0.58) LMNAKDM4EHTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 195 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118084779-A 4-Substituted quinoline amino acid conjugate and preparation method and application thereof 天津科技大学 2024-05-28 CN claimed
US-6903217-B2 Heterocyclylalkylpiperidine derivatives, their preparation and compositions containing them AVENTIS PHARMA S.A. (FR) 2005-06-07 US claimed
US-3989691-A FROM A QUINOLINE PRINCETON UNIVERSITY (US) 1976-11-02 US claimed
US-20260132121-A1 INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF ODYSSEY THERAPEUTICS INC (US) 2026-05-14 US disclosed
US-12624018-B1 Inhibitors of RIPK2 and medical uses thereof ODYSSEY THERAPEUTICS, INC. (US) 2026-05-12 US disclosed
US-12528791-B2 Thyroid hormone receptor beta agonist compounds TERNS PHARMACEUTICALS, INC. (US) 2026-01-20 US disclosed
EP-4622970-A1 INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF ODYSSEY THERAPEUTICS, INC. (US) 2025-10-01 EP disclosed
US-20250059157-A1 TLR7/8 ANTAGONISTS AND USES THEREOF MERCK PATENT GMBH (DE) 2025-02-20 US disclosed
CN-119081100-A FAPi, FAPi intermediate, FAPi modified lipid nanoparticle for encapsulating HSP47 siRNA and application of lipid nanoparticle 华东师范大学 2024-12-06 CN disclosed
US-20240239806-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF TREATING DISORDERS CHENGDU ANTICANCER BIOSCIENCE LTD (CN) 2024-07-18 US disclosed
US-20240239806-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF TREATING DISORDERS CHENGDU ANTICANCER BIOSCIENCE LTD (CN) 2024-07-18 US disclosed
WO-1998022457-A9 ARYL AND HETEROARYL SUBSTITUTED FUSED PYRROLE ANTIINFLAMMATORY AGENTS 1998-08-20 WO disclosed
WO-1998022457-A1 ARYL AND HETEROARYL SUBSTITUTED FUSED PYRROLE ANTIINFLAMMATORY AGENTS AMGEN INC. (US) 1998-05-28 WO disclosed
US-5506235-A Quinoline derivatives as immunostimulants PFIZER INC. (US) 1996-04-09 US disclosed
EP-0597003-A1 QUINOLINE DERIVATIVES AS IMMUNOSTIMULANTS PFIZER INC. (US) 1994-05-18 EP disclosed
EP-0240859-B1 LIPOXYGENASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1993-04-28 EP disclosed
WO-1993003030-A1 QUINOLINE DERIVATIVES AS IMMUNOSTIMULANTS PFIZER INC. (US) 1993-02-18 WO disclosed
US-4761403-A QUINOLONE DERIVATIVES ABBOTT LABORATORIES (US) 1988-08-02 US disclosed
EP-0240859-A2 Lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1987-10-14 EP disclosed
US-3989691-A FROM A QUINOLINE PRINCETON UNIVERSITY (US) 1976-11-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12528791-B2 Thyroid hormone receptor beta agonist compounds THRB, THRA, TSHR LMNA 1704/4885KDM4E 4744/4885HTR1A 267/4885
US-20260132121-A1 INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF RIPK1, RIPK2, RIPK4 LMNA 2558/4885KDM4E 2182/4885HTR1A 3996/4885
US-20240239806-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF TREATING DISORDERS CYP27A1, CPT1A, OAT LMNA 1113/4885KDM4E 4052/4885HTR1A 570/4885
US-20250059157-A1 TLR7/8 ANTAGONISTS AND USES THEREOF TLR7, TLR8, TLR9 LMNA 1762/4885KDM4E 1863/4885HTR1A 813/4885
US-12624018-B1 Inhibitors of RIPK2 and medical uses thereof RIPK2, RIPK1, RIPK4 LMNA 2921/4885KDM4E 3070/4885HTR1A 4442/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.