SCHEMBL15080313

SCHEMBL15080313

CN1C(=O)NC2(CCc3c(Br)cccc3C2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
BACE1 P56817 7/20 0.39
ATM Q13315 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 2/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
ABHD6 Q9BV23 1/20 0.34
PARP10 Q53GL7 1/20 0.33
PARP11 Q9NR21 1/20 0.33
PDE7A Q13946 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7928992 0.79 PDE7A (0.44) PARP10PARP11PDE7A
SCHEMBL12203798 0.77 ALDH1A1 (0.36) ALDH1A1BACE1ATMSMN1; SMN2LMNA
SCHEMBL1814392 0.77 BACE1 (0.51) ALDH1A1BACE1ATMLMNAMAPT
SCHEMBL7917580 0.76 SMN1; SMN2 (0.33) ALDH1A1ATMSMN1; SMN2LMNAMAPT
SCHEMBL7925065 0.75 ADRA2A (0.36) ALDH1A1BACE1ABHD6PARP10PARP11
SCHEMBL14707613 0.74 ABHD6 (0.32) ALDH1A1ABHD6PARP10PARP11PDE7A
SCHEMBL7920070 0.73 ADRA2A (0.34) ABHD6PARP10PARP11PDE7A
SCHEMBL7917831 0.71 PDE7A (0.34) ABHD6PARP10PARP11PDE7A
SCHEMBL15545247 0.70 CES1 (0.41) ABHD6PARP10PARP11
SCHEMBL30421685 0.70 CES1 (0.41) ABHD6PARP10PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8476274-B2 Biaryl spiroaminooxazoline analogues as Alpha2C adrenergic receptor modulators MERCK SHARP & DOHME CORP. (US) 2013-07-02 US disclosed