SCHEMBL15083058

SCHEMBL15083058

Cc1ccc(Cn2c(C)c(C(=O)c3nnc(-c4cccnc4)o3)c3cc(C)ccc32)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
RECQL P46063 1/20 0.44
FAAH O00519 2/20 0.42
CES1 P23141 1/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
KDR P35968 2/20 0.39
GAA P10253 2/20 0.39
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39
EPHB4 P54760 1/20 0.39
PLA2G2A P14555 1/20 0.39
PPARG P37231 2/20 0.39
PTGES2 Q9H7Z7 1/20 0.38
TEK Q02763 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003594 0.96 FAAH (0.47) NPC1RAB9ARECQLFAAHCES1
SCHEMBL2000862 0.89 PTGES2 (0.43) NPC1RAB9ARECQLFAAHCES1
SCHEMBL2006336 0.88 FAAH (0.38) NPC1RAB9ARECQLFAAHCES1
SCHEMBL2008862 0.87 PLA2G2A (0.49) NPC1RAB9AFAAHKDM4EALDH1A1
SCHEMBL2003170 0.86 RAB9A (0.45) NPC1RAB9AFAAHCES1KDM4E
SCHEMBL2002059 0.85 FAAH (0.49) FAAHKDM4EALDH1A1TSHRGAA
SCHEMBL2008741 0.85 PTGES2 (0.44) NPC1RAB9ARECQLFAAHCES1
SCHEMBL2005383 0.85 MAPK1 (0.51) FAAHALDH1A1TSHRGAAMAPT
SCHEMBL2007909 0.84 FAAH (0.48) FAAHALDH1A1TSHRGAAMAPT
SCHEMBL2000438 0.82 FAAH (0.49) FAAHKDM4EALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2610244-A1 Indole compounds Ironwood Pharmaceuticals, Inc. (US) 2013-07-03 EP disclosed