SCHEMBL15083064

SCHEMBL15083064

O=C(O)c1cc(-c2ccnnc2)ns1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.43
STING1 Q86WV6 8/20 0.37
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
HDAC4 P56524 1/20 0.34
WNT3A P56704 4/20 0.33
MAPK14 Q16539 1/20 0.33
ALAD P13716 2/20 0.33
SCD O00767 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15083062 0.83 MAPK14 (0.43) MKNK1MKNK2HDAC4MAPK14
SCHEMBL6843818 0.79 TP53 (0.44)
SCHEMBL2722584 0.79 MKNK1 (0.58) HCAR2MKNK1MKNK2HDAC4
SCHEMBL6740513 0.75 ALAD (0.51) ALAD
SCHEMBL6668534 0.75 ALAD (0.51) ALAD
SCHEMBL28093059 0.75 CA12 (0.49) MAPK14
SCHEMBL26613959 0.73 ATR (0.43) WNT3A
SCHEMBL17208102 0.72 MKNK1 (0.63) HCAR2MKNK1MKNK2HDAC4
SCHEMBL12571313 0.72 DHODH (0.45) HCAR2MKNK1MKNK2HDAC4
SCHEMBL11000258 0.71 ALPL (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8884020-B2 Indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2014-11-11 US disclosed
EP-2610244-A1 Indole compounds Ironwood Pharmaceuticals, Inc. (US) 2013-07-03 EP disclosed