SCHEMBL15085706

SCHEMBL15085706

NC(=O)C1(C(=O)NC2(c3cccc(I)n3)CC2)CC1

nearest known ligand 0.31

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.31
PARP1 P09874 1/20 0.31
PIM1 P11309 1/20 0.31
NPC1 O15118 2/20 0.30
TNF P01375 1/20 0.30
NOD2 Q9HC29 1/20 0.30
NOD1 Q9Y239 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3659466 0.85 ADORA2A (0.34) ADORA2APARP1PIM1NPC1TNF
SCHEMBL15085707 0.83 ADORA2A (0.32) ADORA2A
SCHEMBL3660356 0.77 P2RX7 (0.36) NPC1
SCHEMBL10277612 0.76 NPC1 (0.30) NPC1
SCHEMBL3660006 0.75
SCHEMBL15375625 0.71 NPC1 (0.30) NPC1
SCHEMBL23653854 0.68 FPR2 (0.43) ADORA2APARP1NPC1
SCHEMBL3659469 0.68 ADORA2A (0.35) ADORA2APARP1PIM1
SCHEMBL3659049 0.68 LOXL2 (0.39) PARP1
SCHEMBL3659908 0.64 CHUK (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2445914-B1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-a]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INT (DE) 2015-07-22 EP disclosed
EP-2445909-B1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-a]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INT (DE) 2013-11-13 EP disclosed
US-8481750-B2 Derivatives of 6,7-dihydro-5H-imidazo[1,2-α]imidazole-3-carboxylic acid amides BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-07-09 US disclosed