SCHEMBL1509770

SCHEMBL1509770

CC/C(C)=C(/NC(C)(C)C)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
ALDH1A1 P00352 2/20 0.32
FFAR3 O14843 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11751979 0.77 EPHX1 (0.39) EPHX1ALDH1A1FFAR3
SCHEMBL9447224 0.73 FFAR3 (0.35) ALDH1A1FFAR3TDP1
SCHEMBL9447228 0.73 FFAR3 (0.35) ALDH1A1FFAR3TDP1
SCHEMBL2489029 0.71 EPHX1 (0.45) EPHX1NPC1ALDH1A1ALOX15
SCHEMBL125890 0.70 EPHX1 (0.34) EPHX1KDM4CNPC1MAPTRAB9A
SCHEMBL526285 0.70 EPHX1 (0.34) EPHX1KDM4CNPC1MAPTRAB9A
SCHEMBL1509771 0.70 EPHX1 (0.34) EPHX1KDM4CNPC1MAPTRAB9A
SCHEMBL6356662 0.66
SCHEMBL155565 0.66
Propionic Acid SCHEMBL23467114 0.65 FFAR3 (0.43) KDM4CNPC1MAPTRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4547288-A1 RADIOPAQUE MONOMER AND EMBOLISATION MICROSPHERES COMPRISING SAME Guerbet (FR) 2025-05-07 EP claimed
WO-2024003184-A1 RADIOPAQUE MONOMER AND EMBOLISATION MICROSPHERES COMPRISING SAME GUERBET (FR) 2024-01-04 WO claimed
EP-4299080-A1 RADIO-OPAQUE MONOMER AND EMBOLISATION MICROSPHERES COMPRISING SAME Guerbet (FR) 2024-01-03 EP claimed
US-20230285601-A1 NON DEGRADABLE RADIO-OPAQUE EMBOLISATION MICROSPHERE GUERBET (FR) 2023-09-14 US claimed
US-20230272142-A1 NON-DEGRADABLE EMBOLISATION MICROSPHERE GUERBET (FR) 2023-08-31 US claimed
EP-4041318-A1 NON-DEGRADABLE EMBOLISATION MICROSPHERE Guerbet (FR) 2022-08-17 EP claimed
WO-2021069527-A1 NON-DEGRADABLE EMBOLISATION MICROSPHERE GUERBET (FR) 2021-04-15 WO claimed
EP-2683750-B1 IMPLANTABLE SWELLABLE BIO-RESORBABLE POLYMER OCCLUGEL (FR) 2017-04-19 EP claimed
EP-2683753-B1 IMPLANTABLE BIO-RESORBABLE POLYMER CHARGED WITH FRAGILE MACROMOLECULES OCCLUGEL (FR) 2016-08-03 EP claimed
US-20130344159-A1 IMPLANTABLE SWELLABLE BIO-RESORBABLE POLYMER OCCLUGEL (FR) 2013-12-26 US claimed
US-20120230937-A1 IMPLANTABLE BIO-RESORBABLE POLYMER OCCLUGEL (FR) 2012-09-13 US claimed
WO-2011029867-A1 IMPLANTABLE BIO-RESORBABLE POLYMER OCCLUGEL (FR) 2011-03-17 WO claimed
EP-2295480-A1 Implantable bio-resorbable polymer Occlugel (FR) 2011-03-16 EP claimed
US-12552891-B2 Non-degradable embolisation microsphere GUERBET (FR) 2026-02-17 US disclosed
EP-4547288-A1 RADIOPAQUE MONOMER AND EMBOLISATION MICROSPHERES COMPRISING SAME Guerbet (FR) 2025-05-07 EP disclosed
US-20240018396-A1 LOW TEMPERATURE ACTIVATED RELEASE COATING AND A METHOD OF MAKING 3M INNOVATIVE PROPERTIES COMPANY 2024-01-18 US disclosed
US-5756625-A POLYMER OF C4-C14 ALKYL (METH)ACRYLATE MONOMER AND OPTIONALLY ATLEAST ONE COMONOMER, ALTLEAST ONE VINY UNSATURATED ADDITIVE HAVING BOTH IONIC AND HYDROPHOBIC GROUPS, A SURFACTANT, AND POLYMERIZATION INITIATOR MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1998-05-26 US disclosed
WO-1998016591-A1 STABILIZED ADHESIVE MICROSPHERES MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1998-04-23 WO disclosed
US-5714237-A POLYMER CONTAINING C4-C14 ALKYL (METH)ACRYLATE MONOMERS, INITIATOR, SURFACTANT, AND CHAIN TRANSFER AGENT MINNESOTA MINING MANUFACTURING COMPANY (US) 1998-02-03 US disclosed
WO-1997026286-A1 PARTIALLY CROSS-LINKED MICROSPHERES MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1997-07-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12552891-B2 Non-degradable embolisation microsphere VEGFA, FGB, MSR1 EPHX1 354/4885KDM4C 1703/4885NPC1 2925/4885
US-20130344159-A1 IMPLANTABLE SWELLABLE BIO-RESORBABLE POLYMER CRKL, CMKLR1, BMPR1A EPHX1 1812/4885KDM4C 999/4885NPC1 3962/4885
US-20120230937-A1 IMPLANTABLE BIO-RESORBABLE POLYMER PTH1R, BMP2, BMPR1A EPHX1 2250/4885KDM4C 613/4885NPC1 3728/4885
US-20230285601-A1 NON DEGRADABLE RADIO-OPAQUE EMBOLISATION MICROSPHERE KIT, TIE1, HRH4 EPHX1 170/4885KDM4C 809/4885NPC1 2930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.