SCHEMBL15211565

SCHEMBL15211565

COc1c(OCc2ccc(Cl)cc2Cl)ccc2c(OC(C)=O)c(C)oc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.46
ABCB11 O95342 1/20 0.46
MRGPRX4 Q96LA9 3/20 0.44
ADRB2 P07550 1/20 0.44
FABP3 P05413 1/20 0.44
FABP4 P15090 1/20 0.44
FABP5 Q01469 1/20 0.44
POLB P06746 2/20 0.44
SLC26A4 O43511 1/20 0.44
LMNA P02545 2/20 0.41
HTT P42858 1/20 0.41
S1PR1 P21453 1/20 0.41
S1PR5 Q9H228 1/20 0.41
PTGER1 P34995 2/20 0.41
DUSP3 P51452 1/20 0.40
PTPN5 P54829 1/20 0.40
PTPN11 Q06124 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
SAE1 Q9UBE0 1/20 0.40
UBA2 Q9UBT2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15211259 0.83 HDAC8 (0.47) HDAC8ABCB11MRGPRX4ADRB2FABP3
SCHEMBL15211374 0.80 POLB (0.45) HDAC8ABCB11FABP3FABP4FABP5
SCHEMBL15211549 0.78 SLC26A4 (0.61) POLBSLC26A4MAPTALDH1A1GAA
SCHEMBL15211337 0.78 POLB (0.48) HDAC8MRGPRX4ADRB2FABP3FABP4
SCHEMBL15211265 0.77 SLC26A4 (0.46) HDAC8MRGPRX4ADRB2FABP3FABP4
SCHEMBL15211271 0.75 POLB (0.47) HDAC8MRGPRX4ADRB2FABP3FABP4
SCHEMBL15211631 0.75 MRGPRX4 (0.50) HDAC8MRGPRX4ADRB2FABP3FABP4
SCHEMBL17444916 0.74 HDAC8 (0.48) HDAC8MRGPRX4ADRB2FABP3FABP4
SCHEMBL15211372 0.73 HDAC8 (0.44) HDAC8MRGPRX4ADRB2FABP3FABP4
SCHEMBL17431282 0.73 MRGPRX4 (0.45) HDAC8MRGPRX4ADRB2FABP3FABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2838891-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-02-25 EP disclosed
WO-2013125732-A1 AROMATIC RING COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-08-29 WO disclosed