SCHEMBL15211685

SCHEMBL15211685

CNCC=Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.36
MAPT P10636 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
XPO1 O14980 1/20 0.35
NFE2L2 Q16236 1/20 0.34
AHR P35869 1/20 0.33
PTGS1 P23219 1/20 0.33
APP P05067 1/20 0.33
ACP1 P24666 1/20 0.33
RAPGEF4 Q8WZA2 1/20 0.33
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15211695 0.91 UBE2M (0.35) PPARGPPARDPPARANFE2L2AHR
SCHEMBL15211872 0.91 NFE2L2 (0.38) PPARGPPARDPPARANFE2L2AHR
SCHEMBL15211665 0.89 AHR (0.46) PPARGPPARDPPARAAHRRAPGEF4
SCHEMBL15211460 0.86 CYP1A1 (0.42) AHRPTGS1
SCHEMBL12505799 0.76 IDO1 (0.41) IDO1PPARGPPARDPPARANFE2L2
SCHEMBL2097827 0.75 RPS6KA3 (0.41) IDO1PPARGPPARDPPARANFE2L2
SCHEMBL18187457 0.75 ALDH1A1 (0.42) IDO1PPARGPPARDPPARANFE2L2
SCHEMBL16829586 0.75 IDO1 (0.39) IDO1PPARGPPARDPPARANFE2L2
SCHEMBL16829643 0.75 IDO1 (0.39) IDO1PPARGPPARDPPARANFE2L2
SCHEMBL6553356 0.75 ALDH1A1 (0.42) IDO1PPARGPPARDPPARANFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817312-A1 NOVEL NEUROKININ 1 RECEPTOR ANTAGONIST COMPOUNDS Leo Pharma A/S (DK) 2014-12-31 EP disclosed
WO-2013124286-A1 NOVEL NEUROKININ 1 RECEPTOR ANTAGONIST COMPOUNDS LEO PHARMA A/S (DK) 2013-08-29 WO disclosed