SCHEMBL15211665

SCHEMBL15211665

CNCC=Cc1cc(Cl)cc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AHR P35869 2/20 0.46
RAPGEF4 Q8WZA2 1/20 0.37
SLC13A3 Q8WWT9 1/20 0.33
DDR1 Q08345 3/20 0.33
HTR2A P28223 1/20 0.33
SLC6A4 P31645 1/20 0.33
KCNH2 Q12809 1/20 0.33
NAMPT P43490 1/20 0.32
NOTUM Q6P988 1/20 0.32
ACLY P53396 1/20 0.31
PPARG P37231 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15211685 0.89 IDO1 (0.36) AHRRAPGEF4PPARGPPARDPPARA
SCHEMBL15211695 0.84 UBE2M (0.35) AHRPPARGPPARDPPARA
SCHEMBL15211872 0.84 NFE2L2 (0.38) AHRRAPGEF4HTR2ASLC6A4KCNH2
SCHEMBL256046 0.82 AHR (0.50) AHRRAPGEF4SLC13A3DDR1NOTUM
SCHEMBL15211460 0.79 CYP1A1 (0.42) AHR
SCHEMBL2177901 0.73 AHR (0.55) AHRRAPGEF4SLC13A3NAMPTNOTUM
SCHEMBL16638194 0.72 AHR (0.50) AHRRAPGEF4NOTUM
SCHEMBL20076864 0.71 AHR (0.61) AHR
SCHEMBL27856971 0.69 AHR (0.46) AHRRAPGEF4SLC13A3NOTUM
SCHEMBL16957386 0.69 AHR (0.48) AHRRAPGEF4SLC13A3NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817312-A1 NOVEL NEUROKININ 1 RECEPTOR ANTAGONIST COMPOUNDS Leo Pharma A/S (DK) 2014-12-31 EP disclosed
WO-2013124286-A1 NOVEL NEUROKININ 1 RECEPTOR ANTAGONIST COMPOUNDS LEO PHARMA A/S (DK) 2013-08-29 WO disclosed