SCHEMBL15212365

SCHEMBL15212365

CC(C)(C)C1=NCCc2ccc(N)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.40
NOS2 P35228 2/20 0.40
CES2 O00748 2/20 0.36
TYMS P04818 1/20 0.35
HSD17B10 Q99714 2/20 0.33
CASP1 P29466 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CASP7 P55210 1/20 0.33
PKM P14618 1/20 0.32
RAD52 P43351 1/20 0.32
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
HTR2A P28223 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29554639 1.00 NOS3 (0.40) NOS3NOS2CES2TYMSHSD17B10
SCHEMBL30139746 0.87 HSD17B10 (0.43) NOS3NOS2CES2HSD17B10CASP1
SCHEMBL30014807 0.80 PBRM1 (0.43) CES2TYMSHSD17B10CASP1KDM4E
SCHEMBL7993632 0.77 MAOA (0.50) NOS3NOS2TYMSHSD17B10CASP1
SCHEMBL5775841 0.77 PLAU (0.47) NOS3NOS2CES2TYMSHSD17B10
SCHEMBL30460236 0.76 TYMS (0.38) NOS3NOS2CES2TYMS
SCHEMBL14001394 0.75 NOS3 (0.53) NOS3NOS2HSD17B10KDM4EALDH1A1
SCHEMBL29825835 0.74 CES2 (0.35) NOS3NOS2CES2HSD17B10KDM4E
SCHEMBL11616211 0.74 NOS3 (0.43) NOS3NOS2TYMSHSD17B10CASP1
SCHEMBL31014065 0.72 HRH3 (0.43) SMN1; SMN2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110218235-A A kind of compound and preparation method thereof and application as fluorescence polarization probe in the screening of LXR beta ligands 中山大学 2019-09-10 CN disclosed
EP-2817308-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES AbbVie Inc. (US) 2014-12-31 EP disclosed
WO-2013126656-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES ABBVIE INC. (US) 2013-08-29 WO disclosed