SCHEMBL7993632

SCHEMBL7993632

CC1=NCCc2ccc(N)cc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.50
ALDH1A1 P00352 3/20 0.50
KDM4E B2RXH2 2/20 0.50
MAPT P10636 2/20 0.50
GAA P10253 1/20 0.50
NOS3 P29474 4/20 0.43
NOS2 P35228 3/20 0.43
TYMS P04818 1/20 0.38
CA9 Q16790 1/20 0.36
PDE10A Q9Y233 1/20 0.35
CASP1 P29466 2/20 0.35
HSD17B10 Q99714 2/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CASP7 P55210 1/20 0.35
CRBN Q96SW2 1/20 0.35
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1009906 0.81 MAOA (0.53) MAOAALDH1A1KDM4EMAPTGAA
SCHEMBL1010472 0.78 MAOA (0.50) MAOAALDH1A1KDM4EMAPTGAA
SCHEMBL30656741 0.78 MAOA (0.50) MAOAALDH1A1KDM4EMAPTGAA
SCHEMBL29405492 0.78 MAOA (0.50) MAOAALDH1A1KDM4EMAPTGAA
SCHEMBL11616211 0.78 NOS3 (0.43) MAOAALDH1A1KDM4EMAPTGAA
SCHEMBL1009165 0.78 MAOA (0.50) MAOAALDH1A1KDM4EMAPTGAA
SCHEMBL1011035 0.78 MAOA (0.50) MAOAALDH1A1KDM4EMAPTGAA
SCHEMBL15212365 0.77 NOS3 (0.40) ALDH1A1KDM4EMAPTGAANOS3
SCHEMBL5775841 0.77 PLAU (0.47) ALDH1A1KDM4EMAPTNOS3NOS2
SCHEMBL29554639 0.77 NOS3 (0.40) ALDH1A1KDM4EMAPTGAANOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6277861-B1 FOR TREATMENT AND PROPHYLAXIS OF NERVOUS SYSTEM DISORDERS, PSYCHOLOGICAL DISORDERS, MUSCULAR DISORDERS, DRUG ADDICTION WITHDRAWAL, PAIN SMITHKLINE BEECHAM, P.L.C. (GB) 2001-08-21 US disclosed
EP-0971897-A1 ANTI-CONVULSANT ISOQUINOLYL-BENZAMIDE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 2000-01-19 EP disclosed
WO-1998041507-A1 ANTI-CONVULSANT ISOQUINOLYL-BENZAMIDE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 1998-09-24 WO disclosed