SCHEMBL15280201

SCHEMBL15280201

CCc1ccc(C)c2ccoc12

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.36
KCNA2 P16389 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.33
ESR1 P03372 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
APEX1 P27695 1/20 0.33
MAPK1 P28482 1/20 0.33
ESR2 Q92731 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NQO1 P15559 1/20 0.32
POR P16435 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31
KCNA3 P22001 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28731239 0.82 CYP1A2 (0.34) SMN1; SMN2ESR1TP53POLBAPEX1
SCHEMBL30200194 0.82 CYP1A2 (0.34) SMN1; SMN2ESR1TP53POLBAPEX1
SCHEMBL24946157 0.78 CTRC (0.37) KCNA2GABRA1GABRB2KCNA3
SCHEMBL16381040 0.78 KCNA2 (0.34) KCNA2ESR1ESR2GABRA1GABRB2
SCHEMBL806473 0.78 CYP1A2 (0.39) SMN1; SMN2TP53POLBMAPK1NQO1
SCHEMBL31120928 0.78 CYP1A2 (0.39) SMN1; SMN2TP53POLBMAPK1NQO1
SCHEMBL19297217 0.76 GPR55 (0.36) KCNA2
SCHEMBL15629834 0.74 GAA (0.37) HSD17B10KCNA2POLBMAPK1NQO1
SCHEMBL8750157 0.73 CTRC (0.48) HSD17B10KCNA2TP53POLBMAPK1
SCHEMBL19297064 0.72 LMNA (0.36) HSD17B10SMN1; SMN2POLBMAPK1NQO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616460-B1 HETEROCYCLIC COMPOUNDS FOR TREATING OR PREVENTING DISORDERS CAUSED BY REDUCED NEUROTRANSMISSION OF SEROTONIN, NOREPHNEPHRINE OR DOPAMINE. OTSUKA PHARMA CO LTD (JP) 2015-10-28 EP disclosed
WO-2013137479-A1 DECAHYDROQUINOXALINE DERIVATIVES AND ANALOGS THEREOF OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2013-09-19 WO disclosed