SCHEMBL1531287

SCHEMBL1531287

CC(C)(C)OC(=O)NCCCl

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.58
MEN1 O00255 1/20 0.55
GAA P10253 1/20 0.55
KMT2A Q03164 1/20 0.55
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
CA12 O43570 5/20 0.47
CA1 P00915 5/20 0.47
CA2 P00918 5/20 0.47
CA9 Q16790 5/20 0.47
EPHX1 P07099 1/20 0.47
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
STK17B O94768 1/20 0.42
STK17A Q9UEE5 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GFER P55789 1/20 0.42
IDO1 P14902 2/20 0.41
MALT1 Q9UDY8 1/20 0.41
DRD2 P14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21661235 0.88 TDP1 (0.51) TDP1MEN1GAAKMT2AMAOA
SCHEMBL904060 0.88 TDP1 (0.65) TDP1MEN1GAAKMT2AMAOA
SCHEMBL3341020 0.86 TDP1 (0.67) TDP1MEN1GAAKMT2AMAOA
SCHEMBL8959096 0.86 TDP1 (0.68) TDP1MEN1GAAKMT2AMAOA
SCHEMBL28630680 0.84 TDP1 (0.71) TDP1MEN1GAAKMT2AMAOA
SCHEMBL28636908 0.84 TDP1 (0.71) TDP1MEN1GAAKMT2AMAOA
SCHEMBL1486465 0.84 TDP1 (0.71) TDP1MEN1GAAKMT2AMAOA
SCHEMBL9573730 0.83 TDP1 (0.55) TDP1MEN1GAAKMT2AMAOA
SCHEMBL3020258 0.82 TDP1 (0.81) TDP1MEN1GAAKMT2AMAOA
SCHEMBL569251 0.82 TDP1 (0.74) TDP1MEN1GAAKMT2AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 332 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119080766-B Preparation method and application of fluorescent material based on heterocyclic structure 肇庆创峰高新材料有限公司 2025-01-14 CN claimed
CN-119080766-A Preparation method and application of fluorescent material based on heterocyclic structure 肇庆创峰高新材料有限公司 2024-12-06 CN claimed
CN-112694437-A Preparation method of chlorpheniramine maleate impurity 北京悦康科创医药科技股份有限公司 2021-04-23 CN claimed
CN-108033931-A A kind of synthetic method of N-Boc piperazines 山东铂源药业有限公司 2018-05-15 CN claimed
US-20260007754-A1 Conjugate Molecules DIVERSE BIOTECH INC (US) 2026-01-08 US disclosed
US-20250388602-A1 Tetrahydropyranopyrazole Derivatives for the Treatment of Cancer and Viral Infections GENASE THERAPEUTICS B V (NL) 2025-12-25 US disclosed
EP-4370207-B1 BICYCLIC COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS NIDO BIOSCIENCES INC (US) 2025-12-17 EP disclosed
US-12466829-B2 Spirocyclic piperidine melanocortin subtype-2 receptor (MC2R) antagonists and uses thereof Crinetics Pharmaceuticals, Inc. (US) 2025-11-11 US disclosed
EP-4469461-B1 TETRAHYDROPYRANOPYRAZOLE DERIVATIVES FOR THE TREATMENT OF CANCER AND VIRAL INFECTIONS GENASE THERAPEUTICS B V (NL) 2025-10-15 EP disclosed
US-RE50634-E1 Diaryl macrocycles as modulators of protein kinases Turning Point Therapeutics, Inc. (US) 2025-10-14 US disclosed
EP-4615838-A1 SUBSTITUTED BI-AND TRICYCLIC HSET INHIBITORS Merck Patent GmbH (DE) 2025-09-17 EP disclosed
US-12404281-B2 Diaryl macrocycles as modulators of protein kinases Turning Point Therapeutics, Inc. (US) 2025-09-02 US disclosed
US-5604246-A HAVING POTENCY AGAINST MULTIDRUG RESISTANT TUMORS BOEHRINGER MANNHEIM ITALIA SPA (IT) 1997-02-18 US disclosed
US-5596097-A ANTITUMOR AGENTS THE UNIVERSITY OF VERMONT (US) 1997-01-21 US disclosed
EP-0750619-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA S.p.A. (IT) 1997-01-02 EP disclosed
US-5519029-A ANTITUMOR AGENTS BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1996-05-21 US disclosed
WO-1995024407-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1995-09-14 WO disclosed
EP-0662076-A1 2-AMINOALKYL-5-AMINOALKYLAMINO SUBSTITUTED ISOQUINOINDAZOLE-6-(2H)-ONES WITH ANTITUMOUR ACTIVITY THE UNIVERSITY OF VERMONT (US) 1995-07-12 EP disclosed
CN-1101046-A 2-aminoalkyl-5-aminoalkylamino substituted isoquinoindazole-6(2h)-ones UNIV VERMONT (US) 1995-04-05 CN disclosed
WO-1994006795-A1 2-AMINOALKYL-5-AMINOALKYLAMINO SUBSTITUTED ISOQUINOINDAZOLE-6-(2H)-ONES WITH ANTITUMOUR ACTIVITY THE UNIVERSITY OF VERMONT (US) 1994-03-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12466829-B2 Spirocyclic piperidine melanocortin subtype-2 receptor (MC2R) antagonists and uses thereof MC2R, MC1R, MC3R TDP1 4859/4885MEN1 1173/4885GAA 3392/4885
US-12404281-B2 Diaryl macrocycles as modulators of protein kinases MAP3K20, LCK, MAP3K1 TDP1 1421/4885MEN1 2490/4885GAA 4544/4885
US-20260007754-A1 Conjugate Molecules CD274, PDCD1, PDCD1LG2 TDP1 4187/4885MEN1 2032/4885GAA 2607/4885
US-20250388602-A1 Tetrahydropyranopyrazole Derivatives for the Treatment of Cancer and Viral Infections CCNA1, KRAS, RSU1 TDP1 1804/4885MEN1 364/4885GAA 4077/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.