SCHEMBL15322765

SCHEMBL15322765

O=CC1(c2ncccn2)CC1

nearest known ligand 0.30

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TRIM24 O15164 1/20 0.30
TRIM33 Q9UPN9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4121266 0.74 GRIN1 (0.42)
SCHEMBL23851432 0.70 NFE2L2 (0.33) TRIM24TRIM33
SCHEMBL1255555 0.67 GRIN1 (0.47)
SCHEMBL24608783 0.67 GRIN1 (0.44)
SCHEMBL1255604 0.66 GRIN1 (0.50)
SCHEMBL28635906 0.66 KDM4E (0.32)
SCHEMBL20558313 0.65 CYP19A1 (0.35)
Hydrochloric Acid SCHEMBL2392462 0.65 HSP90AA1 (0.35)
Hydrochloric Acid SCHEMBL667557 0.65 HSP90AA1 (0.35)
SCHEMBL31114034 0.64 VNN1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020085234-A1 MORPHINAN DERIVATIVE 日本ケミファ株式会社 2020-04-30 WO disclosed
EP-2834238-B1 DIACYLGLYCEROL ACYLTRANSFERASE 2 INHIBITORS PFIZER (US) 2017-02-01 EP disclosed
US-9296745-B2 Diacylglycerol acyltransferase 2 inhibitors PFIZER INC. (US) 2016-03-29 US disclosed
US-20150087585-A1 DIACYLGLYCEROL ACYLTRANSFERASE 2 INHIBITORS PFIZER INC. (US) 2015-03-26 US disclosed
EP-2834238-A1 DIACYLGLYCEROL ACYLTRANSFERASE 2 INHIBITORS Pfizer Inc. (US) 2015-02-11 EP disclosed
WO-2013150416-A1 DIACYLGLYCEROL ACYLTRANSFERASE 2 INHIBITORS PFIZER INC. (US) 2013-10-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150087585-A1 DIACYLGLYCEROL ACYLTRANSFERASE 2 INHIBITORS DGAT2, DGAT1, PLAAT2 TRIM24 4029/4885TRIM33 4553/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.