SCHEMBL1532354

SCHEMBL1532354

Cc1cc2nccc(OC(C(=O)O)c3ccccc3)c2cc1F

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 5/20 0.48
PPARG P37231 3/20 0.48
KEAP1 Q14145 7/20 0.45
NFE2L2 Q16236 7/20 0.45
MET P08581 1/20 0.44
KDM4E B2RXH2 1/20 0.42
SRC P12931 2/20 0.37
TGFBR1 P36897 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzene SCHEMBL1532355 0.77 KDM4E (0.46) PPARAPPARGKDM4ESRCTGFBR1
SCHEMBL27294586 0.74 ACHE (0.41) METKDM4ESRCTGFBR1
SCHEMBL21881179 0.69 PPARA (0.68) PPARAPPARGKEAP1NFE2L2KDM4E
SCHEMBL4715482 0.69 MET (0.53) METKDM4E
SCHEMBL21881591 0.67 PPARA (0.74) PPARAPPARGKEAP1NFE2L2KDM4E
SCHEMBL7698955 0.65 PPARA (0.45) PPARAPPARGKDM4ESRC
SCHEMBL21881505 0.64 PPARA (0.56) PPARAPPARGKDM4E
SCHEMBL20045399 0.64 KMT2A (0.51) PPARAPPARG
SCHEMBL20869403 0.64 ALDH1A1 (0.52) PPARAPPARGMETKDM4ESRC
SCHEMBL11397979 0.63 KMT2A (0.64) PPARAPPARGKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4662777-B2 2011-03-30 JP claimed
JP-2006511519-A 2006-04-06 JP claimed
EP-1578423-A1 2-AMINOCARBONYL-QUINOLINE COMPOUNDS AS PLATELET ADENOSINE DIPHOSPHATE RECEPTOR ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 2005-09-28 EP claimed
WO-2004052366-A1 2-AMINOCARBONYL-QUINOLINE COMPOUNDS AS PLATELET ADENOSINE DIPHOSPHATE RECEPTOR ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 2004-06-24 WO claimed
EP-1578423-A1 2-AMINOCARBONYL-QUINOLINE COMPOUNDS AS PLATELET ADENOSINE DIPHOSPHATE RECEPTOR ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 2005-09-28 EP disclosed
WO-2004052366-A1 2-AMINOCARBONYL-QUINOLINE COMPOUNDS AS PLATELET ADENOSINE DIPHOSPHATE RECEPTOR ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 2004-06-24 WO disclosed