SCHEMBL1534035

SCHEMBL1534035

NNC(=O)CCC(N)C(=O)NN

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.44
KDM4E B2RXH2 1/20 0.44
KDM5C P41229 1/20 0.44
PHF8 Q9UPP1 1/20 0.44
KDM2A Q9Y2K7 1/20 0.44
HIF1A Q16665 1/20 0.39
CYP1A2 P05177 2/20 0.38
GRM8 O00222 1/20 0.38
GRM6 O15303 1/20 0.38
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GSR P00390 1/20 0.38
GRIK1 P39086 1/20 0.38
GRM5 P41594 1/20 0.38
GRIA1 P42261 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA3 P42263 1/20 0.38
SLC1A3 P43003 1/20 0.38
SLC1A2 P43004 1/20 0.38
SLC1A1 P43005 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL308629 1.00 CTSD (0.44) CTSDKDM4EKDM5CPHF8KDM2A
SCHEMBL1534041 1.00 CTSD (0.44) CTSDKDM4EKDM5CPHF8KDM2A
SCHEMBL28845044 0.87 CTSD (0.41) CTSDKDM4EKDM5CPHF8KDM2A
SCHEMBL8495405 0.85 ALDH1A1 (0.44) CTSDKDM4EKDM5CPHF8KDM2A
SCHEMBL29833669 0.82 BLM (0.58) HIF1ACYP1A2GRM8GRM6GRIN2D
SCHEMBL288407 0.82 BLM (0.58) HIF1ACYP1A2GRM8GRM6GRIN2D
SCHEMBL10135850 0.82 GSR (0.60) CTSDKDM4EKDM5CPHF8KDM2A
SCHEMBL11215138 0.82 GSR (0.60) CTSDKDM4EKDM5CPHF8KDM2A
SCHEMBL709483 0.82 GRM8 (0.60) KDM4EKDM5CPHF8KDM2ACYP1A2
SCHEMBL709482 0.82 GRM8 (0.60) KDM4EKDM5CPHF8KDM2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 163 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1012208-A4 CROSS-LINKED PARTICLES ACCESS PHARMACEUTICALS AUSTRAL (AU) 2003-06-18 EP claimed
US-6221397-B1 POLYMER CONTAINING REACTIVE GROUPS SELECTED FROM THE GROUP CONSISTING OF CARBOXYL, HYDRAZIDYL, AMINO AND THIOL GROUPS, COVALENTLY LINKED TO A DIHYDRAZIDE SPACER BIOTECH AUSTRALIA PTY LIMITED (AU) 2001-04-24 US claimed
EP-1012208-A1 CROSS-LINKED PARTICLES BIOTECH AUSTRALIA PTY. LIMITED (AU) 2000-06-28 EP claimed
WO-1999011703-A1 CROSS-LINKED PARTICLES BIOTECH AUSTRALIA PTY. LIMITED (US) 1999-03-11 WO claimed
US-5874417-A A CROSSLINKED COMPOSITION HAVING CONJUGATED SITE AT GLUCURONIC ACID WITH A MONO HYDRAZIDE OR A POLYHYDRAZIDE AND A PLURALITY OF CELLS FOR TISSUE ENGINEERING, A COSMETIC AGENT, AND A DRUG; DRUG DELIVERY THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 1999-02-23 US claimed
US-5079155-A Bioaffinity chromatography E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-01-07 US claimed
US-12331197-B2 Power transmission belt DAYCO EUROPE S.R.L. (IT) 2025-06-17 US disclosed
EP-3404056-B1 METHOD FOR PRODUCING THERMOPLASTIC ELASTOMER COMPOSITION ZEON CORP (JP) 2025-06-11 EP disclosed
US-20240350970-A1 SEPARATION FUNCTIONAL LAYER, SEPARATION MEMBRANE, AND METHOD FOR MANUFACTURING SEPARATION FUNCTIONAL LAYER NITTO DENKO CORPORATION (JP) 2024-10-24 US disclosed
US-20240287292-A1 POWER TRANSMISSION BELT DAYCO EUROPE S.R.L. (IT) 2024-08-29 US disclosed
WO-2024166604-A1 SEPARATION FUNCTION LAYER AND SEPARATION MEMBRANE 日東電工株式会社 2024-08-15 WO disclosed
US-20240254346-A1 AQUEOUS PIGMENT DISPERSION FOR PREPARING AQUEOUS INK-JET INK FOR PLASTIC SUBSTRATE, AQUEOUS INK-JET INK, AND PRINTED MATTER DIC CORPORATION (JP) 2024-08-01 US disclosed
US-20240239935-A1 NITRILE GROUP-CONTAINING COPOLYMER RUBBER, RUBBER COMPOSITION AND CROSSLINKED RUBBER ZEON CORPORATION (JP) 2024-07-18 US disclosed
EP-1321481-A1 MODIFIED POLYOLEFIN RESIN, MODIFIED POLYOLEFIN RESIN COMPOSITION, AND USE THEREOF NIPPON PAPER INDUSTRIES CO., LTD. (JP) 2003-06-25 EP disclosed
EP-1012208-A4 CROSS-LINKED PARTICLES ACCESS PHARMACEUTICALS AUSTRAL (AU) 2003-06-18 EP disclosed
US-6221397-B1 POLYMER CONTAINING REACTIVE GROUPS SELECTED FROM THE GROUP CONSISTING OF CARBOXYL, HYDRAZIDYL, AMINO AND THIOL GROUPS, COVALENTLY LINKED TO A DIHYDRAZIDE SPACER BIOTECH AUSTRALIA PTY LIMITED (AU) 2001-04-24 US disclosed
EP-1012208-A1 CROSS-LINKED PARTICLES BIOTECH AUSTRALIA PTY. LIMITED (AU) 2000-06-28 EP disclosed
WO-1999011703-A1 CROSS-LINKED PARTICLES BIOTECH AUSTRALIA PTY. LIMITED (US) 1999-03-11 WO disclosed
EP-0611066-A1 Continuous separation and purification of materials AGRICULTURAL & FOOD RESEARCH COUNCIL (GB) 1994-08-17 EP disclosed
US-5079155-A Bioaffinity chromatography E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-01-07 US disclosed