SCHEMBL15345266

SCHEMBL15345266

NCC(=O)CCC(=O)OC(=O)CCC(=O)CN

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.62
LMNA P02545 1/20 0.62
GABRR1 P24046 1/20 0.55
HTR2C P28335 1/20 0.48
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.35
GLRA1 P23415 1/20 0.33
SLC6A9 P48067 1/20 0.33
OR51E2 Q9H255 1/20 0.33
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27804583 1.00 KDM4E (0.62) KDM4ELMNAGABRR1HTR2CALDH1A1
SCHEMBL5664524 0.95 KDM4E (0.58) KDM4ELMNAGABRR1HTR2CALDH1A1
SCHEMBL28419062 0.91 KDM4E (0.59) KDM4ELMNAGABRR1HTR2CALDH1A1
SCHEMBL28498302 0.89 KDM4E (0.52) KDM4ELMNAGABRR1HTR2CALDH1A1
SCHEMBL27468792 0.87 KDM4E (0.56) KDM4ELMNAGABRR1HTR2CALDH1A1
SCHEMBL28433422 0.85 HTR2C (0.61) KDM4ELMNAGABRR1HTR2CALDH1A1
SCHEMBL367247 0.82 ALDH1A1 (0.48) KDM4ELMNAGABRR1HTR2CALDH1A1
SCHEMBL28900079 0.82 KDM4E (0.50) KDM4ELMNAGABRR1HTR2CALDH1A1
SCHEMBL28842848 0.80 KDM4E (0.44) KDM4ELMNAGABRR1HTR2CALDH1A1
SCHEMBL20658776 0.80 KDM4E (0.48) KDM4ELMNAGABRR1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108472280-A Compounds and methods for treating or preventing hematologic cancers 布罗德研究所股份有限公司 2018-08-31 CN disclosed
CN-107921288-A The targeting conjugate of KSP inhibitor 拜耳医药股份有限公司 2018-04-17 CN disclosed
EP-2657346-B1 METHOD FOR DETECTING CANCER CELL ARKRAY INC (JP) 2017-08-23 EP disclosed
US-9645154-B2 Method for detecting cancer cell ARKRAY, INC. (JP) 2017-05-09 US disclosed
US-20130288273-A1 Method for Detecting Cancer Cell ARKRAY, INC. (JP) 2013-10-31 US disclosed
EP-2657346-A1 METHOD FOR DETECTING CANCER CELL Arkray, Inc. (JP) 2013-10-30 EP disclosed