SCHEMBL15380628

SCHEMBL15380628

O=C(O)c1cccc(C2(C(=O)NC(CN3CCCC3)c3ccccc3)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
MITF O75030 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
GFER P55789 1/20 0.44
PAX8 Q06710 1/20 0.44
ATM Q13315 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
HIF1A Q16665 1/20 0.42
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
OPRK1 P41145 2/20 0.40
MEN1 O00255 1/20 0.40
HSD11B1 P28845 2/20 0.40
GPR88 Q9GZN0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL432280 1.00 ALDH1A1 (0.44) ALDH1A1MITFHTTRAB9AGFER
SCHEMBL10083363 0.92 OPRK1 (0.44) ALDH1A1MITFHTTRAB9AGFER
SCHEMBL432941 0.92 OPRK1 (0.44) ALDH1A1MITFHTTRAB9AGFER
SCHEMBL15385492 0.89 HSD11B1 (0.50) ALDH1A1MITFHTTRAB9AGFER
SCHEMBL435831 0.89 HSD11B1 (0.50) ALDH1A1MITFHTTRAB9AGFER
SCHEMBL10083301 0.88 KMT2A (0.41) ALDH1A1MITFHTTRAB9AGFER
SCHEMBL461186 0.88 ALDH1A1 (0.43) ALDH1A1MITFHTTRAB9AGFER
SCHEMBL15380884 0.88 ALDH1A1 (0.43) ALDH1A1MITFHTTRAB9AGFER
Hydrochloric Acid SCHEMBL15380695 0.88 HSD11B1 (0.49) ALDH1A1MITFHTTRAB9AGFER
Hydrochloric Acid SCHEMBL434246 0.88 HSD11B1 (0.49) ALDH1A1MITFHTTRAB9AGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9303027-B2 Kappa opioid receptor agonists DR. REDDY'S LABORATORIES LTD. (IN) 2016-04-05 US claimed
US-20130303525-A1 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES, INC. (US) 2013-11-14 US claimed
US-9303027-B2 Kappa opioid receptor agonists DR. REDDY'S LABORATORIES LTD. (IN) 2016-04-05 US disclosed
US-20130303525-A1 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES, INC. (US) 2013-11-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130303525-A1 KAPPA OPIOID RECEPTOR AGONISTS OPRK1, OPRL1, OPRD1 ALDH1A1 1649/4885MITF 3668/4885HTT 3363/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.