SCHEMBL15422360

SCHEMBL15422360

C=C(C)C(=O)NC(=O)C=CC

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.35
ALDH1A1 P00352 2/20 0.32
TDP1 Q9NUW8 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15422359 1.00 TGFBR1 (0.35) TGFBR1ALDH1A1TDP1KDM4E
SCHEMBL9550398 0.88 TGFBR1 (0.39) TGFBR1ALDH1A1TDP1KDM4E
SCHEMBL10407850 0.83 ALDH1A1 (0.33) ALDH1A1
SCHEMBL10407848 0.83 ALDH1A1 (0.33) ALDH1A1
SCHEMBL28328511 0.81
SCHEMBL15014686 0.81
SCHEMBL491406 0.80 ALDH1A1 (0.43) TGFBR1ALDH1A1TDP1
SCHEMBL491408 0.80 ALDH1A1 (0.43) TGFBR1ALDH1A1TDP1
SCHEMBL19076272 0.80 ALDH1A1 (0.36) TGFBR1ALDH1A1
SCHEMBL4591815 0.77 ALDH1A1 (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9108923-B2 Compounds, compositions, and methods for cancer therapy HOWARD HUGHES MEDICAL INSTITUTE (US) 2015-08-18 US disclosed
US-20140024639-A1 Compounds, Compositions, and Methods for Cancer Therapy NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2014-01-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140024639-A1 Compounds, Compositions, and Methods for Cancer Therapy MCL1, TP53, VHL TGFBR1 4137/4885ALDH1A1 710/4885TDP1 2640/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.