SCHEMBL15428476

SCHEMBL15428476

CNC[C@@H](Oc1ccc(C(F)(F)F)cc1)[C@H]1CCN(C(=O)O)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
LMNA P02545 4/20 0.41
HRH3 Q9Y5N1 3/20 0.41
NPC1 O15118 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
MTOR P42345 2/20 0.41
RAB9A P51151 2/20 0.41
CYP3A4 P08684 2/20 0.41
SLC6A2 P23975 2/20 0.41
HTR2C P28335 2/20 0.41
SLC6A3 Q01959 2/20 0.41
KDM4E B2RXH2 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9107358 0.89 MMP13 (0.45) ALDH1A1EPHX2
SCHEMBL9107353 0.89 MMP13 (0.45) ALDH1A1EPHX2
SCHEMBL9280632 0.87 LIPC (0.40) SLC6A4HRH3SMYD3EPHX2LIPE
SCHEMBL12468333 0.80 PPARG (0.39) SLC6A4HRH3RAB9ASLC6A2ALDH1A1
SCHEMBL9108211 0.78 MMP13 (0.45) ALDH1A1EPHX2LIPE
SCHEMBL9108220 0.78 MMP13 (0.45) ALDH1A1EPHX2LIPE
SCHEMBL9110045 0.77 DPP4 (0.45) EPHX2
SCHEMBL9110055 0.77 DPP4 (0.45) EPHX2
SCHEMBL14837995 0.76 MMP13 (0.43) EPHX2LIPE
SCHEMBL9281151 0.76 LIPC (0.39) SLC6A4LMNAHRH3CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8637568-B2 Serotonin reuptake inhibitors THERAVANCE, INC. (US) 2014-01-28 US disclosed