SCHEMBL15435554

SCHEMBL15435554

O=CNc1cccnc1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
ALDH1A1 P00352 1/20 0.40
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 2/20 0.40
KDM4E B2RXH2 2/20 0.40
HSP90AA1 P07900 1/20 0.40
IDO1 P14902 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.38
HTT P42858 1/20 0.38
KDM5A P29375 2/20 0.37
PABPC1 P11940 1/20 0.37
MAPT P10636 3/20 0.36
MITF O75030 1/20 0.36
TP53 P04637 1/20 0.36
MAPK10 P53779 1/20 0.36
GFER P55789 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2308076 0.78 TSHR (0.39) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL10430438 0.76 P2RX7 (0.41) TSHRALDH1A1MEN1KMT2ANPSR1
SCHEMBL25043764 0.76 NAPRT (0.41) TSHRALDH1A1MEN1KMT2ARAB9A
SCHEMBL6578328 0.76 BACE1 (0.47) TSHRALDH1A1MEN1KMT2ATDP1
SCHEMBL6589447 0.76 TRIM24 (0.52) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL8763290 0.75 ALDH1A1 (0.57) TSHRALDH1A1MEN1KMT2ANPC1
SCHEMBL30527294 0.75 ALDH1A1 (0.57) TSHRALDH1A1MEN1KMT2ANPC1
SCHEMBL18856198 0.74 PABPC1 (0.43) TSHRALDH1A1MEN1KMT2ANPC1
SCHEMBL1939410 0.74 GAA (0.50) TSHRALDH1A1MEN1KMT2ANPC1
SCHEMBL29876843 0.74 GAA (0.50) TSHRALDH1A1MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2687511-A1 Pyridinone derivatives as tissue transglutaminase inhibitors Zedira GmbH (DE) 2014-01-22 EP disclosed