SCHEMBL154652

SCHEMBL154652

O=c1cnoc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.47
FTO Q9C0B1 3/20 0.47
MAOB P27338 2/20 0.47
CYP3A4 P08684 5/20 0.41
HPGD P15428 5/20 0.41
KDM4E B2RXH2 5/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPT P10636 3/20 0.41
HSD17B10 Q99714 3/20 0.41
GLA P06280 1/20 0.41
PGAM1 P18669 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
CA12 O43570 3/20 0.40
CA1 P00915 3/20 0.40
CA9 Q16790 3/20 0.40
CA2 P00918 2/20 0.40
TNKS O95271 2/20 0.40
PARP1 P09874 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8185680 0.98 MAOA (0.45) MAOAFTOMAOBCYP3A4HPGD
SCHEMBL2005190 0.70 BRD4 (0.41) MAOBSMN1; SMN2CA12CA1CA9
SCHEMBL29917986 0.68 SMN1; SMN2 (0.44) HPGDKDM4ESMN1; SMN2ALDH1A1PARP1
SCHEMBL30411299 0.68 LOXL2 (0.44) HPGDALDH1A1PARP1LMNAMEN1
SCHEMBL928494 0.68 ALDH1A1 (0.50) CYP3A4HPGDKDM4ESMN1; SMN2ALDH1A1
Benzo[D]Isoxazole SCHEMBL8438 0.67
Benzo[D]Isoxazole SCHEMBL1355530 0.67
Benzo[D]Isoxazole SCHEMBL29366929 0.67
SCHEMBL2005193 0.67 BRD4 (0.42) MAOACYP3A4HPGDKDM4ESMN1; SMN2
SCHEMBL24399382 0.65 BRD4 (0.42) MAOBKDM4ESMN1; SMN2ALDH1A1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 774 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025133260-A1 INHIBITORS OF PLASMODIA REMODELING ENZYMES UNIVERSITÄT REGENSBURG, IN VERTRETUNG DES FREISTAATES BAYERN (DE) 2025-06-26 WO claimed
WO-2025099143-A1 COMPOSITIONS FOR STABILIZING POLYMERIC MATERIALS AGAINST UV LIGHT THERMAL AND GAS FADING DEGRADATION CYTEC INDUSTRIES INC. (US) 2025-05-15 WO claimed
WO-2025099141-A1 STABILIZING COMPOSITIONS FOR POLYMERIC MATERIALS CYTEC INDUSTRIES INC. (US) 2025-05-15 WO claimed
CN-117105918-B 1, 4-Benzoxazinone derivative with biological activity and preparation method and application thereof 河南师范大学 2025-03-18 CN claimed
EP-4363506-A1 COMPOSITIONS AND METHODS FOR PROTECTING COATINGS FROM THE DELETERIOUS EFFECTS OF EXPOSURE TO UV-C LIGHT Cytec Industries Inc. (US) 2024-05-08 EP claimed
WO-2024083872-A1 SYNERGISTIC STABILIZER COMPOSITIONS AND METHODS FOR USING SAME FOR PROTECTING ORGANIC MATERIALS FROM UV LIGHT AND THERMAL DEGRADATION CYTEC INDUSTRIES INC. (US) 2024-04-25 WO claimed
CN-117567387-A Method for preparing benzoxazine-4-ketone series compounds by using nitroaromatic hydrocarbon 南京德川医药科技有限公司 2024-02-20 CN claimed
CN-117105918-A 1, 4-benzoxazinone derivative with biological activity and preparation method and application thereof 河南师范大学 2023-11-24 CN claimed
CN-117069711-A Preparation method of benzoxazine-4-one derivative 江苏扬农化工股份有限公司 2023-11-17 CN claimed
WO-2023082029-A1 METHOD FOR PREPARING AN EXTRACT BASED ON ACANTHUS LEAVES (ACANTHUS MOLLIS) AS A NATURAL FUNGICIDE AND INSECTICIDE BUZZETTI MORALES KARINA ANDREA (CL) 2023-05-19 WO claimed
WO-1997048707-A1 4H-3,1-BENZOXAZIN-4-ONE DERIVATIVES AND ANALOGS AS ANTIVIRAL AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-12-24 WO claimed
EP-0674038-B1 Use of 4-H-3,1-benzoxazin-4-one compounds for improving the light fastness of textile materials CLARIANT FINANCE BVI LTD (VG) 1997-10-29 EP claimed
WO-1997035950-A1 BLEACHING POWER ENHANCERS FOR BLEACHES AND TEXTILE WASHING COMPOSITIONS BASF AKTIENGESELLSCHAFT (DE) 1997-10-02 WO claimed
WO-1997035718-A1 STRUCTURE FOR PROTECTING INDIVIDUALS FROM SOLAR ULTRAVIOLET RADIATION POLYMER INNOVATIONS CORPORATION (US) 1997-10-02 WO claimed
EP-0775698-A1 Bis-resorcinol-triazines as UV absorber triazine Ciba SC Holding AG (CH) 1997-05-28 EP claimed
US-5560852-A PRETECTIVE CLOTHING SANDOZ LTD. (CH) 1996-10-01 US claimed
US-5480882-A Benzoxazinone and benzothiazinone derivatives having cardiovascular activity ITALFARMACO S.P.A. (IT) 1996-01-02 US claimed
EP-0606421-A1 DERIVATIVES OF IMIDAZO 5,1-C] 1, 4]BENZOXAZIN-1-ONE AS 5 HT3 ANTAGONISTS PHARMACIA & UPJOHN S.p.A. (IT) 1994-07-20 EP claimed
US-5264539-A Heat resistant films, fibers or moldings with radiation resistance HOECHST CELANESE CORP. (US) 1993-11-23 US claimed
WO-1993021167-A1 THERMALLY STABLE OLIGOMERIC ULTRAVIOLET STABILIZERS HOECHST CELANESE CORPORATION (US) 1993-10-28 WO claimed