SCHEMBL15467947

SCHEMBL15467947

O=C1CNCc2ccc(C(F)(F)F)cc21

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.51
PARP10 Q53GL7 1/20 0.51
TDP2 O95551 2/20 0.47
HTR2A P28223 5/20 0.44
HTR2C P28335 5/20 0.44
HTR2B P41595 5/20 0.44
PNMT P11086 4/20 0.41
ASIC3 Q9UHC3 1/20 0.40
KIF11 P52732 3/20 0.39
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL798153 0.86 TDP2 (0.51) PARP1PARP10TDP2HTR2AHTR2C
SCHEMBL3680946 0.78 PARP1 (0.62) PARP1PARP10TDP2HTR2AHTR2C
SCHEMBL30201259 0.78 PARP1 (0.62) PARP1PARP10TDP2HTR2AHTR2C
SCHEMBL29835145 0.77 PNMT (0.56) PARP1PARP10TDP2HTR2AHTR2C
SCHEMBL2310562 0.77 PNMT (0.56) PARP1PARP10TDP2HTR2AHTR2C
SCHEMBL30681290 0.77 PARP10 (0.71) PARP1PARP10TDP2HTR2AHTR2C
Bromide SCHEMBL2310632 0.76 PNMT (0.54) PARP1PARP10TDP2HTR2AHTR2C
Hydrochloric Acid SCHEMBL29627981 0.76 PNMT (0.54) PARP1PARP10TDP2HTR2AHTR2C
Hydrochloric Acid SCHEMBL1647036 0.76 PNMT (0.54) PARP1PARP10TDP2HTR2AHTR2C
Bromide SCHEMBL2310627 0.74 PNMT (0.53) PARP1PARP10TDP2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8946260-B2 17α-hydroxylase/C17,20-lyase inhibitors NOVARTIS AG (CH) 2015-02-03 US disclosed
US-20140045872-A1 17a-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2014-02-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140045872-A1 17a-HYDROXYLASE/C17,20-LYASE INHIBITORS CYP17A1, CYP21A2, HSD17B1 PARP1 2549/4885PARP10 940/4885TDP2 2986/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.