SCHEMBL15468462

SCHEMBL15468462

CC(=O)Nc1ccc(-c2cnccc2S)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.57
HTT P42858 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
TSHR P16473 2/20 0.49
MAPK10 P53779 1/20 0.47
BRAF P15056 1/20 0.46
KMT2A Q03164 5/20 0.46
MEN1 O00255 3/20 0.46
KDM4E B2RXH2 2/20 0.46
GAA P10253 2/20 0.46
PRNP P04156 1/20 0.46
POLB P06746 1/20 0.46
NISCH Q9Y2I1 1/20 0.46
MAPT P10636 3/20 0.45
HPGD P15428 3/20 0.45
ALDH1A1 P00352 2/20 0.45
RXFP1 Q9HBX9 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15468459 0.79 RPS6KA3 (0.39) SLC22A12SMN1; SMN2TSHRKMT2AMEN1
SCHEMBL28879472 0.78 SLC22A12 (0.56) SLC22A12HTTSMN1; SMN2L3MBTL1TSHR
SCHEMBL29132450 0.78 SMN1; SMN2 (0.60) HTTSMN1; SMN2L3MBTL1KMT2AMEN1
SCHEMBL3728246 0.77 SMN1; SMN2 (0.76) HTTSMN1; SMN2L3MBTL1TSHRMAPK10
SCHEMBL15158977 0.73 SLC22A12 (1.00) SLC22A12
SCHEMBL20020060 0.73 RPS6KA3 (0.68) SLC22A12MAPK10CYP3A4
SCHEMBL11192637 0.73 NPC1 (0.65) HTTSMN1; SMN2L3MBTL1KMT2AKDM4E
SCHEMBL29611891 0.73 NPC1 (0.65) HTTSMN1; SMN2L3MBTL1KMT2AKDM4E
SCHEMBL526972 0.72 POLB (0.60) L3MBTL1KMT2AMEN1KDM4EGAA
SCHEMBL15468461 0.72 LMNA (0.46) SLC22A12MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585437-B1 THIOACETATE COMPOUNDS, COMPOSITIONS AND METHODS OF USE ARDEA BIOSCIENCES INC (US) 2014-02-12 EP disclosed