SCHEMBL20020060

SCHEMBL20020060

Oc1ccc(-c2cnccc2S)cc1

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 6/20 0.68
SLC22A12 Q96S37 2/20 0.45
CYP17A1 P05093 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
ESR1 P03372 3/20 0.39
ESR2 Q92731 2/20 0.39
USP7 Q93009 2/20 0.38
MAPK10 P53779 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15468461 0.83 LMNA (0.46) RPS6KA3SLC22A12CYP3A4
SCHEMBL20020113 0.80 SLC22A12 (0.44) RPS6KA3SLC22A12CYP19A1CYP11B1CYP11B2
SCHEMBL15468467 0.80 SLC22A12 (0.44) RPS6KA3SLC22A12
SCHEMBL30494180 0.76 RPS6KA3 (0.68) RPS6KA3SLC22A12CYP17A1CYP11B1CYP11B2
SCHEMBL11258140 0.76 RPS6KA3 (0.68) RPS6KA3SLC22A12CYP17A1CYP11B1CYP11B2
SCHEMBL16938695 0.76 MAPT (0.55) RPS6KA3SLC22A12CYP3A4
SCHEMBL15468459 0.76 RPS6KA3 (0.39) RPS6KA3SLC22A12CYP17A1CYP3A4
SCHEMBL29153269 0.73 RPS6KA3 (0.70) RPS6KA3SLC22A12CYP17A1CYP3A4CYP19A1
SCHEMBL19955351 0.73 RPS6KA3 (0.63) RPS6KA3SLC22A12CYP19A1CYP11B2ESR1
SCHEMBL15468462 0.73 SLC22A12 (0.57) SLC22A12CYP3A4MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975025-B1 THIOACETATE COMPOUNDS, COMPOSITIONS AND METHODS OF USE ARDEA BIOSCIENCES INC (US) 2018-04-04 EP disclosed