SCHEMBL1549949

SCHEMBL1549949

CCOC(=O)C(F)(C(=O)O)c1ccc(Cl)nn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.38
TSHR P16473 3/20 0.38
ABCB11 O95342 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
HTR2A P28223 1/20 0.38
PMP22 Q01453 1/20 0.38
PPARA Q07869 1/20 0.38
POLB P06746 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 3/20 0.36
MAPT P10636 3/20 0.36
PIN1 Q13526 1/20 0.36
MEN1 O00255 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
KDM4E B2RXH2 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL247624 0.85 KMT2A (0.46) KMT2ATSHRABCB11CYP1A2CYP3A4
SCHEMBL30628250 0.85 KMT2A (0.46) KMT2ATSHRABCB11CYP1A2CYP3A4
SCHEMBL246875 0.84 TSHR (0.40) KMT2ATSHRABCB11CYP1A2CYP3A4
SCHEMBL249487 0.80 CNR2 (0.46) KMT2ATSHRABCB11CYP1A2CYP3A4
SCHEMBL245602 0.80 ABCB11 (0.44) KMT2ATSHRABCB11CYP1A2CYP3A4
SCHEMBL18106959 0.77 LMNA (0.37) KMT2ALMNA
SCHEMBL38656523 0.69 CNR2 (0.41) KMT2ATSHRABCB11CYP1A2CYP3A4
SCHEMBL5764028 0.69 NPSR1 (0.38) KMT2ATSHRABCB11CYP1A2CYP3A4
SCHEMBL5010275 0.67 PIN1 (0.53) KMT2ATSHRPOLBNPSR1LMNA
SCHEMBL1550807 0.67 LMNA (0.41) KMT2ACYP1A2CYP3A4PPARAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2313407-A1 cMET INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2011-04-27 EP disclosed
WO-2010019899-A1 cMET INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed