Roxadimate

Roxadimate

SCHEMBL15518

CCOC(=O)c1ccc(N(CC(C)O)CC(C)O)cc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA7 P43166 2/20 0.53
CA9 Q16790 2/20 0.53
CA14 Q9ULX7 2/20 0.53
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
MAOA P21397 1/20 0.51
RAB9A P51151 6/20 0.49
NPC1 O15118 4/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
TP53 P04637 1/20 0.49
POLB P06746 1/20 0.49
MAPT P10636 4/20 0.47
ALDH1A1 P00352 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Roxadimate SCHEMBL6851586 1.00 CA12 (0.53) CA12CA1CA2CA7CA9
SCHEMBL17576039 0.86 CA12 (0.56) CA12CA1CA2CA7CA9
SCHEMBL25807500 0.84 TSHR (0.49) CA12CA1CA2CA7CA9
SCHEMBL65692 0.82 CA12 (0.61) CA12CA1CA2CA7CA9
SCHEMBL8387891 0.81 CA12 (0.46) CA12CA1CA2CA7CA9
SCHEMBL11570799 0.80 HPGD (0.50) ESR1ESR2LMNARAB9ANPC1
SCHEMBL5065554 0.79 RAB9A (0.47) CA12CA1CA2CA7CA9
SCHEMBL7145665 0.78 TAS2R14 (0.46) CA12CA1CA2CA7CA9
SCHEMBL18387846 0.78 CA1 (0.56) CA12CA1CA2CA7CA9
SCHEMBL2388270 0.78 CA12 (0.56) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4809 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260076889-A1 POLYESTER FILM-FORMING POLYMERS FOR ALCOHOLBASED SUNSCREEN FORMULATIONS NOURYON CHEMICALS INTERNATIONAL B.V. (NL) 2026-03-19 US claimed
US-20250381126-A1 POLYVINYL ALCOHOL FILM-FORMING POLYMERS FOR ALCOHOL-BASED SUNSCREEN FORMULATIONS AND METHODS OF USING SAME NOURYON CHEMICALS INTERNATIONAL B.V. (NL) 2025-12-18 US claimed
US-20250332079-A1 TOPICAL SUNSCREEN CONCEPT MATRIX SOLUTIONS 2025-10-30 US claimed
EP-4577180-A1 POLYESTER FILM-FORMING POLYMERS FOR ALCOHOL-BASED SUNSCREEN FORMULATIONS Nouryon Chemicals International B.V. (NL) 2025-07-02 EP claimed
US-12290590-B2 Biodegradable polyesters for water-resistant anhydrous suncare formulations NOURYON CHEMICALS INTERNATIONAL B.V. (NL) 2025-05-06 US claimed
EP-4543411-A1 POLYVINYL ALCOHOL FILM-FORMING POLYMERS FOR ALCOHOL-BASED SUNSCREEN FORMULATIONS AND METHODS OF USING SAME Nouryon Chemicals International B.V. (NL) 2025-04-30 EP claimed
WO-2024042237-A1 POLYESTER FILM-FORMING POLYMERS FOR ALCOHOL-BASED SUNSCREEN FORMULATIONS NOURYON CHEMICALS INTERNATIONAL B.V. (NL) 2024-02-29 WO claimed
WO-2023247794-A1 POLYVINYL ALCOHOL FILM-FORMING POLYMERS FOR ALCOHOL-BASED SUNSCREEN FORMULATIONS AND METHODS OF USING SAME NOURYON CHEMICALS INTERNATIONAL B.V. (NL) 2023-12-28 WO claimed
CN-116456956-A Solid cosmetic material 株式会社资生堂 2023-07-18 CN claimed
EP-2827835-B2 SUPERABSORBENT POLYMERS AND SILICONE ELASTOMER FOR USE IN SKIN CARE COMPOSITIONS PROCTER & GAMBLE (US) 2022-09-07 EP claimed
CN-1285751-A Antimutagenic compositions for treatment and prevention of photodamage to skin PRO NEURON INC (US) 2001-02-28 CN claimed
EP-1032405-A1 ANTIMUTAGENIC COMPOSITIONS FOR TREATMENT AND PREVENTION OF PHOTODAMAGE TO SKIN PRO-NEURON, INC. (US) 2000-09-06 EP claimed
US-5976555-A EMULSIFIER SYSTEM JOHNSON & JOHNSON CONSUMER PRODUCTS, INC. (US) 1999-11-02 US claimed
WO-1999022741-A1 ANTIMUTAGENIC COMPOSITIONS FOR TREATMENT AND PREVENTION OF PHOTODAMAGE TO SKIN PRO-NEURON, INC. (US) 1999-05-14 WO claimed
EP-0885000-A2 TOPICAL COMPOSITIONS COMPRISING AN OIL-IN-WATER EMULSION AND A RETINOID Johnson & Johnson Consumer Companies, Inc. (US) 1998-12-23 EP claimed
WO-1997031620-A2 TOPICAL COMPOSITIONS COMPRISING AN OIL-IN-WATER EMULSION AND A RETINOID JOHNSON & JOHNSON CONSUMER PRODUCTS, INC. (US) 1997-09-04 WO claimed
US-5567420-A SUCH AS SUNSCREEN AGENT GE CANADA FINANCE HOLDING COMPANY (CA) 1996-10-22 US claimed
WO-1996014826-A1 LOTION WHICH IS TEMPORARILY COLORED UPON APPLICATION SEEUV (US) 1996-05-23 WO claimed
WO-1996014053-A1 SKIN CLEANSING - UV SCREENING COMPOSITION CUSSONS (INTERNATIONAL) LIMITED (GB) 1996-05-17 WO claimed
US-4293544-A SUNSCREEN AGENTS FINETEX INCORPORATED (US) 1981-10-06 US claimed