Roxadimate

Roxadimate

SCHEMBL6851586

CCOC(=O)c1ccc(N(CC(C)O)CC(C)O)cc1.CCOC(=O)c1ccc(N(CC(C)O)CC(C)O)cc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA7 P43166 2/20 0.53
CA9 Q16790 2/20 0.53
CA14 Q9ULX7 2/20 0.53
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
MAOA P21397 1/20 0.51
RAB9A P51151 6/20 0.49
NPC1 O15118 4/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
TP53 P04637 1/20 0.49
POLB P06746 1/20 0.49
MAPT P10636 4/20 0.47
ALDH1A1 P00352 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Roxadimate SCHEMBL15518 1.00 CA12 (0.53) CA12CA1CA2CA7CA9
SCHEMBL17576039 0.86 CA12 (0.56) CA12CA1CA2CA7CA9
SCHEMBL25807500 0.84 TSHR (0.49) CA12CA1CA2CA7CA9
SCHEMBL65692 0.82 CA12 (0.61) CA12CA1CA2CA7CA9
SCHEMBL8387891 0.81 CA12 (0.46) CA12CA1CA2CA7CA9
SCHEMBL11570799 0.80 HPGD (0.50) ESR1ESR2LMNARAB9ANPC1
SCHEMBL5065554 0.79 RAB9A (0.47) CA12CA1CA2CA7CA9
SCHEMBL7145665 0.78 TAS2R14 (0.46) CA12CA1CA2CA7CA9
SCHEMBL18387846 0.78 CA1 (0.56) CA12CA1CA2CA7CA9
SCHEMBL2388270 0.78 CA12 (0.56) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1423371-A1 TRIAZINE DERIVATIVES AND THEIR USE AS SUNSCREENS Ciba SC Holding AG (CH) 2004-06-02 EP disclosed
WO-2003016289-A1 TRIAZINE DERIVATIVES AND THEIR USE AS SUNSCREENS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2003-02-27 WO disclosed